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2-(Isopropylamino)thieno[3,2-d]pyrimidin-4(3H)-one derivatives as selective phosphodiesterase 7 inhibitors with potent in vivo efficacy
by
Endo, Yusuke
,
Kawai, Kentaro
,
Asano, Takeshi
,
Amano, Seiji
,
Asanuma, Yoshihito
,
Sawada, Keisuke
,
Onodera, Yuuta
,
Ueo, Noriko
,
Takahashi, Nobuaki
,
Sonoda, Yo
,
Kamei, Noriyuki
,
Irie, Tetsumi
Published in
Bioorganic & medicinal chemistry letters
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Bioorganic & Medicinal Chemistry Letters
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Animals
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Anti-Inflammation
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Aqueous Solubility
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Chemistry
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Chemistry, Medicinal
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Chemistry, Organic
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Cyclic Nucleotide Phosphodiesterases, Type 7 - Antagonists & Inhibitors
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Cyclic Nucleotide Phosphodiesterases, Type 7 - Metabolism
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Disease Models, Animal
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Dose-Response Relationship, Drug
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Edema - Chemically Induced
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Edema - Drug Therapy
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Life Sciences & Biomedicine
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Male
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Mice
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Mice, Inbred Icr
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Molecular Structure
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Pharmacology & Pharmacy
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Phorbol Esters
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Sciencedirect®
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Sciencedirect Journals
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Backfile Package - Organic Chemistry (Legacy) [Yco]
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