5‑Fluoroindole Reduces the Bacterial Burden in a Murine Model of Mycobacterium tuberculosis Infection by Neves, Christiano E., Paz, Josiane D., Abbadi, Bruno L., Rambo, Raoní S., Czeczot, Alexia M., Sperotto, Nathalia D. M., Dadda, Adilio S., Silva, Rodrigo B. M., Perelló, Marcia A., Gonçalves, Guilherme A., González, Laura C., Bizarro, Cristiano V., Machado, Pablo, Basso, Luiz A.

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Synthesis and Antimycobacterial Activity of 3-Phenyl-1H-indoles by Jardim Etchart, Renata, Rambo, Raoní S., Lopes Abbadi, Bruno, Sperotto, Nathalia, Ev Neves, Christiano, Fries Silva, Fernanda, Dornelles, Maiele, Duarte, Lovaine, Souza Macchi, Fernanda, Alberton Perelló, Marcia, Vescia Lourega, Rogério, Valim Bizarro, Cristiano, Basso, Luiz Augusto, Machado, Pablo

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Crystal structure of dihydroneopterin aldolase from Mycobacterium tuberculosis associated with 8-mercaptoguanine, and development of novel S8-functionalized analogues as inhibitors... by Czeczot, Alexia de Matos, Muniz, Mauro Neves, Perelló, Marcia Alberton, Silva, Éverton Edésio Dinis, Timmers, Luís Fernando Saraiva Macedo, Berger, Andresa, Gonzalez, Laura Calle, Arraché Gonçalves, Guilherme, Moura, Sidnei, Machado, Pablo, Bizarro, Cristiano Valim, Basso, Luiz Augusto

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Exploring Scaffold Hopping for Novel 2‑(Quinolin-4-yloxy)acetamides with Enhanced Antimycobacterial Activity by Borsoi, Ana Flávia, Silva Ramos, Alessandro, Sperotto, Nathalia, Abbadi, Bruno Lopes, Souza Macchi Hopf, Fernanda, da Silva Dadda, Adilio, Scheibler Rambo, Raoní, Neves Muniz, Mauro, Delgado Paz, Josiane, Silveira Grams, Estevão, Fries da Silva, Fernanda, Pissinate, Kenia, Galina, Luiza, Calle González, Laura, Silva Duarte, Lovaine, Alberton Perelló, Marcia, de Matos Czeczot, Alexia, Bizarro, Cristiano Valim, Basso, Luiz Augusto, Machado, Pablo

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Antitubercular Activity of Novel 2‑(Quinoline-4-yloxy)acetamides with Improved Drug-Like Properties by Borsoi, Ana Flávia, Alice, Laura Manzoli, Sperotto, Nathalia, Ramos, Alessandro Silva, Abbadi, Bruno Lopes, Macchi Hopf, Fernanda Souza, Silva Dadda, Adilio da, Rambo, Raoní S., Madeira Silva, Rodrigo Braccini, Paz, Josiane Delgado, Pissinate, Kenia, Muniz, Mauro Neves, Neves, Christiano Ev, Galina, Luiza, González, Laura Calle, Perelló, Marcia Alberton, de Matos Czeczot, Alexia, Leyser, Mariana, de Oliveira, Sílvia Dias, de Araújo Lock, Graziela, de Araújo, Bibiana Verlindo, Costa, Teresa Dalla, Bizarro, Cristiano Valim, Basso, Luiz Augusto, Machado, Pablo

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Synthesis and Antimycobacterial Evaluation of N -(4-(Benzyloxy)benzyl)-4-aminoquinolines by Grams, Estevão Silveira, Silva Ramos, Alessandro, Neves Muniz, Mauro, Rambo, Raoní S, Alberton Perelló, Marcia, Sperotto, Nathalia, Calle González, Laura, Duarte, Lovaine Silva, Galina, Luiza, Silva Dadda, Adilio, Arraché Gonçalves, Guilherme, Valim Bizarro, Cristiano, Basso, Luiz Augusto, Machado, Pablo

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Unveiling the Antimycobacterial Potential of Novel 4-Alkoxyquinolines: Insights into Selectivity, Mechanism of Action, and In Vivo Exposure by da Silva, Fernanda Fries, Paz, Josiane Delgado, Rambo, Raoní Scheibler, Gonçalves, Guilherme Arraché, Muniz, Mauro Neves, de Matos Czeczot, Alexia, Perelló, Marcia Alberton, Berger, Andresa, González, Laura Calle, Duarte, Lovaine Silva, da Silva, Anelise Baptista, Ferreira, Carlos Alexandre Sanchez, de Oliveira, Sílvia Dias, Moura, Sidnei, Bizarro, Cristiano Valim, Basso, Luiz Augusto, Machado, Pablo

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Novel 4-aminoquinolines: Synthesis, inhibition of the Mycobacterium tuberculosis enoyl-acyl carrier protein reductase, antitubercular activity, SAR, and preclinical evaluation by Paz, Josiane Delgado, Denise de Moura Sperotto, Nathalia, Ramos, Alessandro Silva, Pissinate, Kenia, da Silva Rodrigues Junior, Valnês, Abbadi, Bruno Lopes, Borsoi, Ana Flávia, Rambo, Raoní Scheibler, Corso Minotto, Ana Carolina, da Silva Dadda, Adilio, Galina, Luiza, Macchi Hopf, Fernanda Souza, Muniz, Mauro Neves, Borges Martinelli, Leonardo Kras, Roth, Candida Deves, Madeira Silva, Rodrigo Braccini, Perelló, Marcia Alberton, de Matos Czeczot, Alexia, Neves, Christiano Ev, Duarte, Lovaine Silva, Leyser, Mariana, Dias de Oliveira, Sílvia, Bizarro, Cristiano Valim, Machado, Pablo, Basso, Luiz Augusto

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Identification of potential inhibitors of Mycobacterium tuberculosis shikimate kinase: molecular docking, in silico toxicity and in vitro experiments by Freitas de Freitas, Talita, Roth, Candida Deves, Abbadi, Bruno Lopes, Hopf, Fernanda Souza Macchi, Perelló, Marcia Alberton, de Matos Czeczot, Alexia, de Souza, Eduardo Vieira, Borsoi, Ana Flávia, Machado, Pablo, Bizarro, Cristiano Valim, Basso, Luiz Augusto, Timmers, Luis Fernando Saraiva Macedo

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Identification of antimycobacterial 8-hydroxyquinoline derivatives as in vitro enzymatic inhibitors of Mycobacterium tuberculosis enoyl-acyl carrier protein reductase by Joaquim, Angélica Rocha, Lopes, Marcela Silva, Fortes, Isadora Serraglio, de Bem Gentz, Caroline, de Matos Czeczot, Alexia, Perelló, Marcia Alberton, Roth, Candida Deves, Vainstein, Marilene Henning, Basso, Luiz Augusto, Bizarro, Cristiano Valim, Machado, Pablo, de Andrade, Saulo Fernandes

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Targeting thymidine phosphorylase inhibition in human colorectal cancer xenografts by Sperotto, Nathalia D. de Moura, Silva, Rodrigo Braccini Madeira, Perelló, Marcia Alberton, Borsoi, Ana Flávia, da Silva Dadda, Adilio, Roth, Candida Deves, Freitas, Raquel Dal Sasso, de Souza, Ana Paula Duarte, Freitas, Deise do Nascimento de, Picada, Jaqueline Nascimento, de Sousa, Jayne Torres, Nabinger, Débora Dreher, Altenhofen, Stefani, Bonan, Carla Denise, Rodrigues-Junior, Valnês S., Bizarro, Cristiano Valim, Basso, Luiz Augusto, Machado, Pablo

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Identification and characterization of new structural scaffolds modulating the activity of Mycobacterium tuberculosis dihydroneopterin aldolase (FolB) in vitro by Virginia Carla de Almeida Falcão, Alexia de Matos Czeczot, Alexia de Matos Czeczot, Mohammad Maqusood Alam, Kyu-Ho Paul Park, Jinyeong Heo, Minjeong Woo, Ana Micaela Camini, Luis Fernando Saraiva Macedo Timmers, Luis Fernando Saraiva Macedo Timmers, Luis Fernando Saraiva Macedo Timmers, David Shum, Marcia Alberton Perelló, Luiz Augusto Basso, Luiz Augusto Basso, Luiz Augusto Basso, Pablo Machado, Pablo Machado, Pablo Machado, Cristiano Valim Bizarro, Cristiano Valim Bizarro, Vincent Delorme

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Evaluation of 3-Deoxy-D-Arabino-Heptulosonate 7-Phosphate Synthase (DAHPS) as a Vulnerable Target in Mycobacterium tuberculosis by Galina, Luiza, Hopf, Fernanda S. M., Abbadi, Bruno Lopes, Sperotto, Nathalia D. de Moura, Czeczot, Alexia M., Duque-Villegas, Mario A., Perello, Marcia Alberton, Matter, Letícia Beatriz, de Souza, Eduardo Vieira, Parish, Tanya, Machado, Pablo, Basso, Luiz A., Bizarro, Cristiano V.

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EPSP Synthase-Depleted Cells Are Aromatic Amino Acid Auxotrophs in Mycobacterium smegmatis by Duque-Villegas, Mario Alejandro, Abbadi, Bruno Lopes, Romero, Paulo Ricardo, Matter, Letícia Beatriz, Galina, Luiza, Dalberto, Pedro Ferrari, Rodrigues-Junior, Valnês da Silva, Ducati, Rodrigo Gay, Roth, Candida Deves, Rambo, Raoní Scheibler, de Souza, Eduardo Vieira, Perello, Marcia Alberton, Morbidoni, Héctor Ricardo, Machado, Pablo, Basso, Luiz Augusto, Bizarro, Cristiano Valim

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