Discovery of GS-9131: Design, synthesis and optimization of amidate prodrugs of the novel nucleoside phosphonate HIV reverse transcriptase (RT) inhibitor GS-9148 by Mackman, Richard L., Ray, Adrian S., Hui, Hon C., Zhang, Lijun, Birkus, Gabriel, Boojamra, Constantine G., Desai, Manoj C., Douglas, Janet L., Gao, Ying, Grant, Deborah, Laflamme, Genevieve, Lin, Kuei-Ying, Markevitch, David Y., Mishra, Ruchika, McDermott, Martin, Pakdaman, Rowchanak, Petrakovsky, Oleg V., Vela, Jennifer E., Cihlar, Tomas

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Design, synthesis, and anti-HIV activity of 4′-modified carbocyclic nucleoside phosphonate reverse transcriptase inhibitors by Boojamra, Constantine G., Parrish, Jay P., Sperandio, David, Gao, Ying, Petrakovsky, Oleg V., Lee, Sharon K., Markevitch, David Y., Vela, Jennifer E., Laflamme, Genevieve, Chen, James M., Ray, Adrian S., Barron, Abraham C., Sparacino, Mark L., Desai, Manoj C., Kim, Choung U., Cihlar, Tomas, Mackman, Richard L.

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Chalcomycin Biosynthesis Gene Cluster from Streptomyces bikiniensis: Novel Features of an Unusual Ketolide Produced through Expression of the chm Polyketide Synthase in Streptomyce... by WARD, Shannon L, ZHIHAO HU, SCHIRMER, Andreas, REID, Ralph, REVILL, W. Peter, REEVES, Christopher D, PETRAKOVSKY, Oleg V, DONG, Steven D, KATZ, Leonard

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Synthesis and anti-HIV activity of 2′-fluorine modified nucleoside phosphonates: Analogs of GS-9148 by Mackman, Richard L., Lin, Kuei-Ying, Boojamra, Constantine G., Hui, Hon, Douglas, Janet, Grant, Deborah, Petrakovsky, Oleg, Prasad, Vidya, Ray, Adrian S., Cihlar, Tomas

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Synthesis, anti-HIV activity, and resistance profiles of ribose modified nucleoside phosphonates by Mackman, Richard L., Boojamra, Constantine G., Prasad, Vidya, Zhang, Lijun, Lin, Kuei-Ying, Petrakovsky, Oleg, Babusis, Darius, Chen, James, Douglas, Janet, Grant, Deborah, Hui, Hon C., Kim, Choung U., Markevitch, David Y., Vela, Jennifer, Ray, Adrian, Cihlar, Tomas

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