SAT182 Effects Of An Orally Bioavailable Nonpeptide Parathyroid Hormone Receptor Type 1 (PTH1R) Antagonist In Rodent Models Of Primary Hyperparathyroidism (PHPT) by Antwan, Agnes S, Rico-Bautista, Elizabeth, Pontillo, Joe, Wang, Shimiao, Johns, Michael, Ramms, Bastian, Fowler, Melissa A, Nguyen, Julie B, Castellanos Gonzalez, Anel A, Fleck, Beth, Retting, Kelsey, Dalvie, Deepak, Betz, Stephen F, Markison, Stacy

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Potent and orally active non-peptide antagonists of the human melanocortin-4 receptor based on a series of trans-2-disubstituted cyclohexylpiperazines by Tucci, Fabio C., White, Nicole S., Markison, Stacy, Joppa, Margaret, Tran, Joe A., Fleck, Beth A., Madan, Ajay, Dyck, Brian P., Parker, Jessica, Pontillo, Joseph, Melissa Arellano, L., Marinkovic, Dragan, Jiang, Wanlong, Chen, Caroline W., Gogas, Kathleen R., Goodfellow, Val S., Saunders, John, Foster, Alan C., Chen, Chen

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4-{(2R)-[3-Aminopropionylamido]-3-(2,4-dichlorophenyl)propionyl}-1-{2-[(2-thienyl)ethylaminomethyl]phenyl}piperazine as a Potent and Selective Melanocortin-4 Receptor AntagonistDe... by Chen, Pontillo, Joseph, Fleck, Beth A, Gao, Yinghong, Wen, Jenny, Tran, Joe A, Tucci, Fabio C, Marinkovic, Dragan, Foster, Alan C, Saunders, John

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Optimization of piperazinebenzylamines with a N-(1-methoxy-2-propyl) side chain as potent and selective antagonists of the human melanocortin-4 receptor by Pontillo, Joseph, Marinkovic, Dragan, Tran, Joe A., Arellano, Melissa, Fleck, Beth A., Wen, Jenny, Tucci, Fabio C., Nelson, Jodie, Saunders, John, Foster, Alan C., Chen, Chen

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Identification of agonists and antagonists of the human melanocortin-4 receptor from piperazinebenzylamines by Tran, Joe A., Pontillo, Joseph, Arellano, Melissa, White, Nicole S., Fleck, Beth A., Marinkovic, Dragan, Tucci, Fabio C., Lanier, Marion, Nelson, Jodie, Saunders, John, Foster, Alan C., Chen, Chen

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Structure–activity relationship studies on a series of cyclohexylpiperazines bearing a phanylacetamide as ligands of the human melanocortin-4 receptor by Pontillo, Joseph, Tran, Joe A., White, Nicole S., Arellano, Melissa, Fleck, Beth A., Marinkovic, Dragan, Tucci, Fabio C., Saunders, John, Foster, Alan C., Chen, Chen

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Arylpropionylpiperazines as antagonists of the human melanocortin-4 receptor by Jiang, Wanlong, Tucci, Fabio C., Chen, Caroline W., Arellano, Melissa, Tran, Joe A., White, Nicole S., Marinkovic, Dragan, Pontillo, Joseph, Fleck, Beth A., Wen, Jenny, Saunders, John, Madan, Ajay, Foster, Alan C., Chen, Chen

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Pyrrolidinones as orally bioavailable antagonists of the human melanocortin-4 receptor with anti-cachectic activity by Tran, Joe A., Tucci, Fabio C., Jiang, Wanlong, Marinkovic, Dragan, Chen, Caroline W., Arellano, Melissa, Markison, Stacy, Fleck, Beth A., Wen, Jenny, White, Nicole S., Pontillo, Joseph, Saunders, John, Marks, Daniel, Hoare, Sam R., Madan, Ajay, Foster, Alan C., Chen, Chen

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Propionylpiperazines as human melanocortin-4 receptor ligands by Chen, Caroline W., Tran, Joe A., Jiang, Wanlong, Tucci, Fabio C., Arellano, Melissa, Wen, Jenny, Fleck, Beth A., Marinkovic, Dragan, White, Nicole S., Pontillo, Joseph, Saunders, John, Madan, Ajay, Foster, Alan C., Chen, Chen

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Design, synthesis, and SAR studies on a series of 2-pyridinylpiperazines as potent antagonists of the melanocortin-4 receptor by Tran, Joe A., Pontillo, Joseph, Fleck, Beth A., Marinkovic, Dragan, Arellano, Melissa, Tucci, Fabio C., Lanier, Marion, Saunders, John, Jiang, Wanlong, Chen, Caroline W., Foster, Alan C., Chen, Chen

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4-{( 2R )-[3-Aminopropionylamido]-3-(2,4-dichlorophenyl)propionyl}-1-{2-[(2-thienyl)ethylaminomethyl]phenyl}piperazine as a Potent and Selective Melanocortin-4 Receptor AntagonistD... by Chen, Pontillo, Joseph, Fleck, Beth A., Gao, Yinghong, Wen, Jenny, Tran, Joe A., Tucci, Fabio C., Marinkovic, Dragan, Foster, Alan C., Saunders, John

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