Discovery of Novel Human Constitutive Androstane Receptor Agonists with the Imidazo[1,2‑a]pyridine Structure by Mejdrová, Ivana, Dušek, Jan, Škach, Kryštof, Stefela, Alžbeta, Skoda, Josef, Chalupský, Karel, Dohnalová, Klára, Pavkova, Ivona, Kronenberger, Thales, Rashidian, Azam, Smutná, Lucie, Duchoslav, Vojtěch, Smutny, Tomas, Pávek, Petr, Nencka, Radim

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Inhibition of FLT3-ITD Kinase in Acute Myeloid Leukemia by New Imidazo[1,2‑b]pyridazine Derivatives Identified by Scaffold Hopping by Břehová, Petra, Řezníčková, Eva, Škach, Kryštof, Jorda, Radek, Dejmek, Milan, Vojáčková, Veronika, Šála, Michal, Kovalová, Markéta, Dračínský, Martin, Dolníková, Alexandra, Strmeň, Timotej, Kinnertová, Monika, Chalupský, Karel, Dvořáková, Alexandra, Gucký, Tomáš, Mertlíková Kaiserová, Helena, Klener, Pavel, Nencka, Radim, Kryštof, Vladimír

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PF74 and Its Novel Derivatives Stabilize Hexameric Lattice of HIV-1 Mature-Like Particles by Dostálková, Alžběta, Škach, Kryštof, Kaufman, Filip, Křížová, Ivana, Hadravová, Romana, Flegel, Martin, Ruml, Tomáš, Hrabal, Richard, Rumlová, Michaela

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Exploring positions 6 and 7 of a quinazoline-based scaffold leads to changes in selectivity and potency towards RIPK2/3 kinases by Misehe, Mbilo, Matoušová, Marika, Dvořáková, Alexandra, Hercík, Kamil, Škach, Kryštof, Chalupská, Dominika, Dejmek, Milan, Šála, Michal, Hájek, Miroslav, Boura, Evzen, Mertlíková-Kaiserová, Helena, Nencka, Radim

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A simple, high-throughput stabilization assay to test HIV-1 uncoating inhibitors by Dostálková, Alžběta, Hadravová, Romana, Kaufman, Filip, Křížová, Ivana, Škach, Kryštof, Flegel, Martin, Hrabal, Richard, Ruml, Tomáš, Rumlová, Michaela

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Structure–activity relationship study of small-molecule inhibitor of Atg12-Atg3 protein–protein interaction by Skach, Krystof, Boserle, Jiri, Nuta, Gal Chaim, Břehová, Petra, Bialik, Shani, Carvalho, Silvia, Kozer, Noga, Barr, Haim, Chaloupecká, Ema, Kimchi, Adi, Nencka, Radim

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