Discovery of Potent, Highly Selective, and In Vivo Efficacious, Allosteric MALT1 Inhibitors by Iterative Scaffold Morphing by Pissot Soldermann, Carole, Simic, Oliver, Renatus, Martin, Erbel, Paulus, Melkko, Samu, Wartmann, Markus, Bigaud, Marc, Weiss, Andreas, McSheehy, Paul, Endres, Ralf, Santos, Paulo, Blank, Jutta, Schuffenhauer, Ansgar, Bold, Guido, Buschmann, Nicole, Zoller, Thomas, Altmann, Eva, Manley, Paul W, Dix, Ina, Buchdunger, Elisabeth, Scesa, Julien, Quancard, Jean, Schlapbach, Achim, Bornancin, Frédéric, Radimerski, Thomas, Régnier, Catherine H

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Discovery of Ligands for TRIM58, a Novel Tissue-Selective E3 Ligase by Hoegenauer, Klemens, An, Shaojian, Axford, Jake, Benander, Christina, Bergsdorf, Christian, Botsch, Josephine, Chau, Suzanne, Fernández, César, Gleim, Scott, Hassiepen, Ulrich, Hunziker, Juerg, Joly, Emilie, Keller, Aramis, Lopez Romero, Sandra, Maher, Robert, Mangold, Anne-Sophie, Mickanin, Craig, Mihalic, Manuel, Neuner, Philippe, Patterson, Andrew W., Perruccio, Francesca, Roggo, Silvio, Scesa, Julien, Schröder, Martin, Shkoza, Dojna, Thai, Binh, Vulpetti, Anna, Renatus, Martin, Reece-Hoyes, John S.

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Discovery and SAR of potent, orally available 2,8-diaryl-quinoxalines as a new class of JAK2 inhibitors by Pissot-Soldermann, Carole, Gerspacher, Marc, Furet, Pascal, Gaul, Christoph, Holzer, Philipp, McCarthy, Clive, Radimerski, Thomas, Regnier, Catherine H., Baffert, Fabienne, Drueckes, Peter, Tavares, Gisele A., Vangrevelinghe, Eric, Blasco, Francesca, Ottaviani, Giorgio, Ossola, Flavio, Scesa, Julien, Reetz, Janitha

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