Image-Based Annotation of Chemogenomic Libraries for Phenotypic Screening by Tjaden, Amelie, Chaikuad, Apirat, Kowarz, Eric, Marschalek, Rolf, Knapp, Stefan, Schröder, Martin, Müller, Susanne

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Therapeutic targeting of p300/CBP HAT domain for the treatment of NUT midline carcinoma by Zhang, Xin, Zegar, Tim, Lucas, Anais, Morrison-Smith, Chevaun, Knox, Tatiana, French, Christopher A., Knapp, Stefan, Müller, Susanne, Siveke, Jens T.

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Progress towards a public chemogenomic set for protein kinases and a call for contributions by Drewry, David H, Wells, Carrow I, Andrews, David M, Angell, Richard, Al-Ali, Hassan, Axtman, Alison D, Capuzzi, Stephen J, Elkins, Jonathan M, Ettmayer, Peter, Frederiksen, Mathias, Gileadi, Opher, Gray, Nathanael, Hooper, Alice, Knapp, Stefan, Laufer, Stefan, Luecking, Ulrich, Michaelides, Michael, Müller, Susanne, Muratov, Eugene, Denny, R Aldrin, Saikatendu, Kumar S, Treiber, Daniel K, Zuercher, William J, Willson, Timothy M

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Discovery and Optimization of Small-Molecule Ligands for the CBP/p300 Bromodomains by Hay, Duncan A, Fedorov, Oleg, Martin, Sarah, Singleton, Dean C, Tallant, Cynthia, Wells, Christopher, Picaud, Sarah, Philpott, Martin, Monteiro, Octovia P, Rogers, Catherine M, Conway, Stuart J, Rooney, Timothy P. C, Tumber, Anthony, Yapp, Clarence, Filippakopoulos, Panagis, Bunnage, Mark E, Müller, Susanne, Knapp, Stefan, Schofield, Christopher J, Brennan, Paul E

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3,5-Dimethylisoxazoles Act As Acetyl-lysine-mimetic Bromodomain Ligands by Hewings, David S, Wang, Minghua, Philpott, Martin, Fedorov, Oleg, Uttarkar, Sagar, Filippakopoulos, Panagis, Picaud, Sarah, Vuppusetty, Chaitanya, Marsden, Brian, Knapp, Stefan, Conway, Stuart J, Heightman, Tom D

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Testis specific gene expression drives disease progression and Rituximab resistance in lymphoma by Knapp, Stefan

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Large-Scale Structural Analysis of the Classical Human Protein Tyrosine Phosphatome by Barr, Alastair J., Ugochukwu, Emilie, Lee, Wen Hwa, King, Oliver N.F., Filippakopoulos, Panagis, Alfano, Ivan, Savitsky, Pavel, Burgess-Brown, Nicola A., Müller, Susanne, Knapp, Stefan

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Comparative structural analyses of the NHL domains from the human E3 ligase TRIM-NHL family by Chaikuad, Apirat, Zhubi, Rezart, Tredup, Claudia, Knapp, Stefan

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A comparison of protein kinases inhibitor screening methods using both enzymatic activity and binding affinity determination by Rudolf, Amalie Frederikke, Skovgaard, Tine, Knapp, Stefan, Jensen, Lars Juhl, Berthelsen, Jens

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PFI-1, a Highly Selective Protein Interaction Inhibitor, Targeting BET Bromodomains by PICAUD, Sarah, DA COSTA, David, BRADNER, James E, TANIERE, Philippe, O'SULLIVAN, Brendan, MÜLLER, Susanne, SCHWALLER, Juerg, STANKOVIC, Tatjana, KNAPP, Stefan, THANASOPOULOU, Angeliki, FILIPPAKOPOULOS, Panagis, FISH, Paul V, PHILPOTT, Martin, FEDOROV, Oleg, BRENNAN, Paul, BUNNAGE, Mark E, OWEN, Dafydd R

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Discovery of a Chemical Tool Inhibitor Targeting the Bromodomains of TRIM24 and BRPF by Bennett, James, Fedorov, Oleg, Tallant, Cynthia, Monteiro, Octovia, Meier, Julia, Gamble, Vicky, Savitsky, Pavel, Nunez-Alonso, Graciela A, Haendler, Bernard, Rogers, Catherine, Brennan, Paul E, Müller, Susanne, Knapp, Stefan

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Chemogenomics for NR1 nuclear hormone receptors by Isigkeit, Laura, Schallmayer, Espen, Busch, Romy, Brunello, Lorene, Menge, Amelie, Elson, Lewis, Müller, Susanne, Knapp, Stefan, Stolz, Alexandra, Marschner, Julian A., Merk, Daniel

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Structure of the Bone Morphogenetic Protein Receptor ALK2 and Implications for Fibrodysplasia Ossificans Progressiva by Chaikuad, Apirat, Alfano, Ivan, Kerr, Georgina, Sanvitale, Caroline E., Boergermann, Jan H., Triffitt, James T., von Delft, Frank, Knapp, Stefan, Knaus, Petra, Bullock, Alex N.

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Discovery of Novel Small-Molecule Inhibitors of BRD4 Using Structure-Based Virtual Screening by Vidler, Lewis R, Filippakopoulos, Panagis, Fedorov, Oleg, Picaud, Sarah, Martin, Sarah, Tomsett, Michael, Woodward, Hannah, Brown, Nathan, Knapp, Stefan, Hoelder, Swen

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LP99: Discovery and Synthesis of the First Selective BRD7/9 Bromodomain Inhibitor by Clark, Peter G. K., Vieira, Lucas C. C., Tallant, Cynthia, Fedorov, Oleg, Singleton, Dean C., Rogers, Catherine M., Monteiro, Octovia P., Bennett, James M., Baronio, Roberta, Müller, Susanne, Daniels, Danette L., Méndez, Jacqui, Knapp, Stefan, Brennan, Paul E., Dixon, Darren J.

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Alternative splicing promotes tumour aggressiveness and drug resistance in African American prostate cancer by Wang, Bi-Dar, Ceniccola, Kristin, Hwang, SuJin, Andrawis, Ramez, Horvath, Anelia, Freedman, Jennifer A., Olender, Jacqueline, Knapp, Stefan, Ching, Travers, Garmire, Lana, Patel, Vyomesh, Garcia-Blanco, Mariano A., Patierno, Steven R., Lee, Norman H.

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New opportunities for kinase drug repurposing and target discovery by Knapp, Stefan

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SH2 domains: modulators of nonreceptor tyrosine kinase activity by Filippakopoulos, Panagis, Müller, Susanne, Knapp, Stefan

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Chemoproteomics and Chemical Probes for Target Discovery by Drewes, Gerard, Knapp, Stefan

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Inhibition of bromodomain and extra-terminal proteins targets constitutively active NFκB and STAT signaling in lymphoma and influences the expression of the antiapoptotic proteins... by Pieper, Nadja M, Schnell, Julia, Bruecher, Daniela, Knapp, Stefan, Vogler, Meike

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