RGS6, RGS7, RGS9, and RGS11 Stimulate GTPase Activity of Gi Family G-proteins with Differential Selectivity and Maximal Activity by Hooks, Shelley B, Waldo, Gary L, Corbitt, James, Bodor, Erik T, Krumins, Andrejs M, Harden, T Kendall

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Mechanism of Phosphorylation-induced Activation of Phospholipase C-γ Isozymes by Gresset, Aurelie, Hicks, Stephanie N., Harden, T. Kendall, Sondek, John

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UDP Is a Competitive Antagonist at the Human P2Y14 Receptor by Fricks, Ingrid P, Maddileti, Savitri, Carter, Rhonda L, Lazarowski, Eduardo R, Nicholas, Robert A, Jacobson, Kenneth A, Harden, T Kendall

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Virtual screening leads to the discovery of novel non-nucleotide P2Y1 receptor antagonists by Costanzi, Stefano, Santhosh Kumar, T., Balasubramanian, Ramachandran, Kendall Harden, T., Jacobson, Kenneth A.

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Synthesis of extended uridine phosphonates derived from an allosteric P2Y2 receptor ligand by Song, Lijun, Risseeuw, Martijn D P, Karalic, Izet, Barrett, Matthew O, Brown, Kyle A, Harden, T Kendall, Van Calenbergh, Serge

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Induction of Novel Agonist Selectivity for the ADP-Activated P2Y1 Receptor Versus the ADP-Activated P2Y12 and P2Y13 Receptors by Conformational Constraint of an ADP Analog by Chhatriwala, Mariya, Ravi, R Gnana, Patel, Roshni I, Boyer, Jose L, Jacobson, Kenneth A, Harden, T Kendall

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A selective high-affinity antagonist of the P2Y14 receptor inhibits UDP-glucose-stimulated chemotaxis of human neutrophils by Barrett, Matthew O, Sesma, Juliana I, Ball, Christopher B, Jayasekara, P Suresh, Jacobson, Kenneth A, Lazarowski, Eduardo R, Harden, T Kendall

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Quantitation of extracellular UTP using a sensitive enzymatic assay by Lazarowski, Eduardo R, Harden, T Kendall

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P2Y1 Antagonists:  Combining Receptor-Based Modeling and QSAR for a Quantitative Prediction of the Biological Activity Based on Consensus Scoring by Costanzi, Stefano, Tikhonova, Irina G, Ohno, Michihiro, Roh, Eun Joo, Joshi, Bhalchandra V, Colson, Anny-Odile, Houston, Dayle, Maddileti, Savitri, Harden, T. Kendall, Jacobson, Kenneth A

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Purification and Functional Reconstitution of the Human P2Y12 Receptor by Bodor, Erik T, Waldo, Gary L, Hooks, Shelley B, Corbitt, James, Boyer, Jose L, Harden, T Kendall

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A membrane-associated, fluorogenic reporter for mammalian phospholipase C isozymes by Huang, Weigang, Wang, Xiaoyang, Endo-Streeter, Stuart, Barrett, Matthew, Waybright, Jarod, Wohlfeld, Christian, Hajicek, Nicole, Harden, T. Kendall, Sondek, John, Zhang, Qisheng

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General and Versatile Autoinhibition of PLC Isozymes by Hicks, Stephanie N., Jezyk, Mark R., Gershburg, Svetlana, Seifert, Jason P., Harden, T. Kendall, Sondek, John

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Regulation of P2Y1 Receptor-Mediated Signaling by the Ectonucleoside Triphosphate Diphosphohydrolase Isozymes NTPDase1 and NTPDase2 by Alvarado-Castillo, Claudia, Harden, T Kendall, Boyer, José L

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Loss of P2Y1 receptor desensitization does not impact hemostasis or thrombosis despite increased platelet reactivity in vitro by Paul, David S., Blatt, Tasha N., Schug, Wyatt J., Clark, Emily G., Kawano, Tomohiro, Mackman, Nigel, Murcia, Sebastian, Poe, Kathryn O., Mwiza, Jean Marie N., Harden, T. Kendall, Bergmeier, Wolfgang, Nicholas, Robert A.

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Enigmatic GPCR finds a stimulating drug by Harden, T Kendall

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Molecular dynamics simulation of the P2Y14 receptor. Ligand docking and identification of a putative binding site of the distal hexose moiety by IVANOV, Andrei A, FRICKS, Ingrid, KENDALL HARDEN, T, JACOBSON, Kenneth A

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Quantitation of the P2Y1 Receptor with a High Affinity Radiolabeled Antagonist by Waldo, Gary L., Corbitt, James, Boyer, José L., Ravi, Gnana, Kim, Hak Sung, Ji, Xiao-Duo, Lacy, James, Jacobson, Kenneth A., Harden, T. Kendall

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Synthesis and P2Y2 receptor agonist activities of uridine 5′-phosphonate analogues by Van Poecke, Sara, Barrett, Matthew O., Santhosh Kumar, T., Sinnaeve, Davy, Martins, José C., Jacobson, Kenneth A., Kendall Harden, T., Van Calenbergh, Serge

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Mechanisms of release of nucleotides and integration of their action as P2X- and P2Y-receptor activating molecules by Lazarowski, Eduardo R, Boucher, Richard C, Harden, T Kendall

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Agonist Versus Antagonist Action of ATP at the P2Y4 Receptor Is Determined by the Second Extracellular Loop by Herold, Christopher L., Qi, Ai-Dong, Harden, T. Kendall, Nicholas, Robert A.

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