Design, Synthesis, SAR, and Biological Evaluation of Highly Potent Benzimidazole-Spaced Phosphono-α-Amino Acid Competitive NMDA Antagonists of the AP-6 Type by Baudy, Reinhardt B, Yardley, John P, Zaleska, Margaret M, Bramlett, Donna R, Tasse, Rene P, Kowal, Dianne M, Katz, Alan H, Moyer, John A, Abou-Gharbia, Magid

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Design and Synthesis of [2-(8,9-Dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)- ethyl]phosphonic Acid (EAA-090), a Potent N-Methyl-d-aspartate Antagonist, via the Use of 3-Cyclobut... by Kinney, William A, Abou-Gharbia, Magid, Garrison, Deanna T, Schmid, Jean, Kowal, Dianne M, Bramlett, Donna R, Miller, Tracy L, Tasse, Rene P, Zaleska, Margaret M, Moyer, John A

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Bioisosteric replacement of the .alpha.-amino carboxylic acid functionality in 2-amino-5-phosphonopentanoic acid yields unique 3,4-diamino-3-cyclobutene-1,2-dione containing NMDA a... by Kinney, William A, Lee, Nancy E, Garrison, Deanna T, Podlesny, Edward J, Simmonds, Joanne T, Bramlett, Donna, Notvest, Ronald R, Kowal, Dianne M, Tasse, Rene P

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A [ 35S]GTP γS binding assessment of metabotropic glutamate receptor standards in Chinese hamster ovary cell lines expressing the human metabotropic receptor subtypes 2 and 4 by Kowal, Dianne, Hsiao, Chu-Lai, Ge, Albert, Wardwell-Swanson, Judith, Ghosh, Krishnendu, Tasse, Rene

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Discovery of a highly potent, functionally-selective muscarinic M1 agonist, way-132983 using rational drug design and receptor modelling by SABB, A. L, HUSBANDS, G. M, TOKOLICS, J, STEIN, R. P, TASSE, R. P, BOAST, C. A, MOYER, J. A, ABOU-GHARBIA, M

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Design and models for estimating antagonist potency (pA 2, Kd and IC 50) following the detection of antagonism observed in the presence of intrinsic activity by Ghosh, Krishnendu, Kowal, Dianne, Dawson, Lee A., Tasse, Rene

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Discovery of a highly potent, functionally-selective muscarinic M 1 agonist,WAY-132983 using rational drug design and receptor modelling by Sabb, Annmarie L., Husbands, G.Morris, Tokolics, Joseph, Stein, Reinhardt P., Tasse, Rene P., Boast, Carl A., Moyer, John A., Abou-Gharbia, Magid

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Potent quinoxaline-spaced phosphono .alpha.-amino acids of the AP-6 type as competitive NMDA antagonists: synthesis and biological evaluation by Baudy, Reinhardt B, Greenblatt, Lynne P, Jirkovsky, Ivo L, Conklin, Mary, Russo, Ralph J, Bramlett, Donna R, Emrey, Tracy A, Simmonds, Joanne T, Kowal, Dianne M

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Neuroprotective interaction effects of NMDA and AMPA receptor antagonists in an in vitro model of cerebral ischemia by Arias, Robert L, Tasse, J.René P, Bowlby, Mark R

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WAY-131256 is an orally active, efficacious, and in vivo functionally selective M1 agonist by Sabb, Annmarie L., Stein, Reinhardt P., Vogel, Robert L., Tasse, Rene, Amburn, Susan, Fairman, Denise K., Kowal, Dianne, Malhotra, Deepa, Boast, Carl A., Bartolomeo, Adam, Morris, Herman, Sailer, Tracy, Moyer, John A., Abou-Gharbia, Magid, Ho, Douglas M.

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Potency Difference between the Zwitterion Form and the Cation Forms of Tetrodotoxin by Camougis, George, Takman, Bertil H., J. Rene P. Tasse

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Electrographic Studies of Cardiac Activity of the Cladoceran, Daphnia by Tasse, J. Rene P, Camougis, George

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Electrographic Studies of Cardiac Activity of the Cladoceran, Daphnia by Camougis, George, Tasse, J. René P.

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