Combined Use of Crystalline Sodium Salt and Polymeric Precipitation Inhibitors to Improve Pharmacokinetic Profile of Ibuprofen through Supersaturation by Terebetski, Jenna L., Cummings, John J., Fauty, Scott E., Michniak-Kohn, Bozena

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Combining ibuprofen sodium with cellulosic polymers: A deep dive into mechanisms of prolonged supersaturation by Terebetski, Jenna L., Michniak-Kohn, Bozena

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Discovery of MK-3168: A PET Tracer for Imaging Brain Fatty Acid Amide Hydrolase by Liu, Ping, Hamill, Terence G, Chioda, Marc, Chobanian, Harry, Fung, Selena, Guo, Yan, Chang, Linda, Bakshi, Raman, Hong, Qingmei, Dellureficio, James, Lin, Linus S, Abbadie, Catherine, Alexander, Jessica, Jin, Hong, Mandala, Suzanne, Shiao, Lin-Lin, Li, Wenping, Sanabria, Sandra, Williams, David, Zeng, Zhizhen, Hajdu, Richard, Jochnowitz, Nina, Rosenbach, Mark, Karanam, Bindhu, Madeira, Maria, Salituro, Gino, Powell, Joyce, Xu, Ling, Terebetski, Jenna L, Leone, Joseph F, Miller, Patricia, Cook, Jacquelynn, Holahan, Marie, Joshi, Aniket, O’Malley, Stacey, Purcell, Mona, Posavec, Diane, Chen, Tsing-Bau, Riffel, Kerry, Williams, Mangay, Hargreaves, Richard, Sullivan, Kathleen A, Nargund, Ravi P, DeVita, Robert J

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Fragment-based lead discovery of a novel class of small molecule antagonists of neuropeptide B/W receptor subtype 1 (GPR7) by Moningka, Remond, Romero, F. Anthony, Hastings, Nicholas B., Guo, Zhiqiang, Wang, Ming, Di Salvo, Jerry, Li, Ying, Trusca, Dorina, Deng, Qiaoling, Tong, Vincent, Terebetski, Jenna L., Ball, Richard G., Ujjainwalla, Feroze

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Discovery of phenyl acetamides as potent and selective GPR119 agonists by Zhu, Cheng, Wang, Liping, Zhu, Yuping, Guo, Zack Zhiqiang, Liu, Ping, Hu, Zhiyong, Szewczyk, Jason W., Kang, Ling, Chicchi, Gary, Ehrhardt, Anka, Woods, Andrea, Seo, Toru, Woods, Morgan, van Heek, Margaret, Dingley, Karen H., Pang, Jianmei, Salituro, Gino M., Powell, Joyce, Terebetski, Jenna L., Hornak, Viktor, Campeau, Louis-Charles, Orr, Robert K., Ujjainwalla, Feroze, Miller, Michael, Stamford, Andrew, Wood, Harold B., Kowalski, Timothy, Nargund, Ravi P., Edmondson, Scott D.

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Discovery of MK-4409, a Novel Oxazole FAAH Inhibitor for the Treatment of Inflammatory and Neuropathic Pain by Chobanian, Harry R, Guo, Yan, Liu, Ping, Chioda, Marc D, Fung, Selena, Lanza, Thomas J, Chang, Linda, Bakshi, Raman K, Dellureficio, James P, Hong, Qingmei, McLaughlin, Mark, Belyk, Kevin M, Krska, Shane W, Makarewicz, Amanda K, Martel, Elliot J, Leone, Joseph F, Frey, Lisa, Karanam, Bindhu, Madeira, Maria, Alvaro, Raul, Shuman, Joyce, Salituro, Gino, Terebetski, Jenna L, Jochnowitz, Nina, Mistry, Shruti, McGowan, Erin, Hajdu, Richard, Rosenbach, Mark, Abbadie, Catherine, Alexander, Jessica P, Shiao, Lin-Lin, Sullivan, Kathleen M, Nargund, Ravi P, Wyvratt, Matthew J, Lin, Linus S, DeVita, Robert J

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Design of Potent and Orally Active GPR119 Agonists for the Treatment of Type II Diabetes by Liu, Ping, Hu, Zhiyong, DuBois, Byron G, Moyes, Christopher R, Hunter, David N, Zhu, Cheng, Kar, Nam Fung, Zhu, Yuping, Garfunkle, Joie, Kang, Ling, Chicchi, Gary, Ehrhardt, Anka, Woods, Andrea, Seo, Toru, Woods, Morgan, van Heek, Margaret, Dingley, Karen H, Pang, Jianmei, Salituro, Gino M, Powell, Joyce, Terebetski, Jenna L, Hornak, Viktor, Campeau, Louis-Charles, Lamberson, Joe, Ujjainwalla, Fez, Miller, Michael, Stamford, Andrew, Wood, Harold B, Kowalski, Timothy, Nargund, Ravi P, Edmondson, Scott D

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Improved Stability of Proline-Derived Direct Thrombin Inhibitors through Hydroxyl to Heterocycle Replacement by Chobanian, Harry R, Pio, Barbara, Guo, Yan, Shen, Hong, Huffman, Mark A, Madeira, Maria, Salituro, Gino, Terebetski, Jenna L, Ormes, James, Jochnowitz, Nina, Hoos, Lizbeth, Zhou, Yuchen, Lewis, Dale, Hawes, Brian, Mitnaul, Lyndon, O’Neill, Kim, Ellsworth, Kenneth, Wang, Liangsu, Biftu, Tesfaye, Duffy, Joseph L

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The discovery of potent antagonists of NPBWR1 (GPR7) by Anthony Romero, F., Hastings, Nicholas B., Moningka, Remond, Guo, Zhiqiang, Wang, Ming, Di Salvo, Jerry, Lei, Ying, Trusca, Dorina, Deng, Qiaolin, Tong, Vincent, Terebetski, Jenna L., Ball, Richard G., Ujjainwalla, Feroze

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Inhaled formulation and device selection: bridging the gap between preclinical species and first-in-human studies by Wylie, Jennifer L, House, Aileen, Mauser, Peter J, Sellers, Shari, Terebetski, Jenna, Wang, Zhenyu, Ehrick, Jason D

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Discovery and Optimization of a Novel Triazole Series of GPR142 Agonists for the Treatment of Type 2 Diabetes by Guo, Liangqin, Parker, Dann L, Zang, Yi, Sweis, Ramzi F, Liu, Weiguo, Sherer, Edward C, Buist, Nicole, Terebetski, Jenna, Kelly, Terri, Bugianesi, Randal, Priest, Birgit T, Dingley, Karen H, Li, Xiaofang, Mitelman, Stan, Salituro, Gino, Trujillo, Maria E, Pachanski, Michele, Kirkland, Melissa, Powles, Mary Ann, Eiermann, George J, Feng, Yue, Shang, Jin, Howard, Andrew D, Ujjainwalla, Feroze, Sinz, Christopher J, Debenham, John S, Edmondson, Scott D, Nargund, Ravi P, Hagmann, William K, Li, Derun

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