Multistage and transmission-blocking targeted antimalarials discovered from the open-source MMV Pandemic Response Box by Reader, Janette, van der Watt, Mariëtte E., Taylor, Dale, Le Manach, Claire, Mittal, Nimisha, Ottilie, Sabine, Theron, Anjo, Moyo, Phanankosi, Erlank, Erica, Nardini, Luisa, Venter, Nelius, Lauterbach, Sonja, Bezuidenhout, Belinda, Horatscheck, Andre, van Heerden, Ashleigh, Spillman, Natalie J., Cowell, Anne N., Connacher, Jessica, Opperman, Daniel, Orchard, Lindsey M., Llinás, Manuel, Istvan, Eva S., Goldberg, Daniel E., Boyle, Grant A., Calvo, David, Mancama, Dalu, Coetzer, Theresa L., Winzeler, Elizabeth A., Duffy, James, Koekemoer, Lizette L., Basarab, Gregory, Chibale, Kelly, Birkholtz, Lyn-Marié

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Nowhere to hide: interrogating different metabolic parameters of Plasmodium falciparum gametocytes in a transmission blocking drug discovery pipeline towards malaria elimination by Reader, Janette, Botha, Mariëtte, Theron, Anjo, Lauterbach, Sonja B, Rossouw, Claire, Engelbrecht, Dewaldt, Wepener, Melanie, Smit, Annél, Leroy, Didier, Mancama, Dalu, Coetzer, Theresa L, Birkholtz, Lyn-Marie

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In vitro anti-malarial interaction and gametocytocidal activity of cryptolepine by Forkuo, Arnold Donkor, Ansah, Charles, Mensah, Kwesi Boadu, Annan, Kofi, Gyan, Ben, Theron, Anjo, Mancama, Dalu, Wright, Colin W

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Open Source Drug Discovery with the Malaria Box Compound Collection for Neglected Diseases and Beyond by Van Voorhis, Wesley C, Adams, John H, Adelfio, Roberto, Ahyong, Vida, Akabas, Myles H, Alano, Pietro, Alday, Aintzane, Alemán Resto, Yesmalie, Alsibaee, Aishah, Alzualde, Ainhoa, Andrews, Katherine T, Avery, Simon V, Avery, Vicky M, Ayong, Lawrence, Baker, Mark, Baker, Stephen, Ben Mamoun, Choukri, Bhatia, Sangeeta, Bickle, Quentin, Bounaadja, Lotfi, Bowling, Tana, Bosch, Jürgen, Boucher, Lauren E, Boyom, Fabrice F, Brea, Jose, Brennan, Marian, Burton, Audrey, Caffrey, Conor R, Camarda, Grazia, Carrasquilla, Manuela, Carter, Dee, Belen Cassera, Maria, Chih-Chien Cheng, Ken, Chindaudomsate, Worathad, Chubb, Anthony, Colon, Beatrice L, Colón-López, Daisy D, Corbett, Yolanda, Crowther, Gregory J, Cowan, Noemi, D'Alessandro, Sarah, Le Dang, Na, Delves, Michael, DeRisi, Joseph L, Du, Alan Y, Duffy, Sandra, Abd El-Salam El-Sayed, Shimaa, Ferdig, Michael T, Fernández Robledo, José A, Fidock, David A, Florent, Isabelle, Fokou, Patrick V T, Galstian, Ani, Gamo, Francisco Javier, Gokool, Suzanne, Gold, Ben, Golub, Todd, Goldgof, Gregory M, Guha, Rajarshi, Guiguemde, W Armand, Gural, Nil, Guy, R Kiplin, Hansen, Michael A E, Hanson, Kirsten K, Hemphill, Andrew, Hooft van Huijsduijnen, Rob, Horii, Takaaki, Horrocks, Paul, Hughes, Tyler B, Huston, Christopher, Igarashi, Ikuo, Ingram-Sieber, Katrin, Itoe, Maurice A, Jadhav, Ajit, Naranuntarat Jensen, Amornrat, Jensen, Laran T, Jiang, Rays H Y, Kaiser, Annette, Keiser, Jennifer, Ketas, Thomas, Kicka, Sebastien, Kim, Sunyoung, Kirk, Kiaran, Kumar, Vidya P, Kyle, Dennis E, Lafuente, Maria Jose, Landfear, Scott, Lee, Nathan, Lee, Sukjun, Lehane, Adele M, Li, Fengwu, Little, David, Liu, Liqiong, Llinás, Manuel, Loza, Maria I, Lubar, Aristea, Lucantoni, Leonardo, Lucet, Isabelle, Maes, Louis, Mancama, Dalu

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Identification and Profiling of a Novel Diazaspiro[3.4]octane Chemical Series Active against Multiple Stages of the Human Malaria Parasite Plasmodium falciparum and Optimization Ef... by Le Manach, Claire, Dam, Jean, Woodland, John G, Kaur, Gurminder, Khonde, Lutete P, Brunschwig, Christel, Njoroge, Mathew, Wicht, Kathryn J, Horatscheck, André, Paquet, Tanya, Boyle, Grant A, Gibhard, Liezl, Taylor, Dale, Lawrence, Nina, Yeo, Tomas, Mok, Sachel, Eastman, Richard T, Dorjsuren, Dorjbal, Talley, Daniel C, Guo, Hui, Simeonov, Anton, Reader, Janette, van der Watt, Mariëtte, Erlank, Erica, Venter, Nelius, Zawada, Jacek W, Aswat, Ayesha, Nardini, Luisa, Coetzer, Theresa L, Lauterbach, Sonja B, Bezuidenhout, Belinda C, Theron, Anjo, Mancama, Dalu, Koekemoer, Lizette L, Birkholtz, Lyn-Marie, Wittlin, Sergio, Delves, Michael, Ottilie, Sabine, Winzeler, Elizabeth A, von Geldern, Thomas W, Smith, Dennis, Fidock, David A, Street, Leslie J, Basarab, Gregory S, Duffy, James, Chibale, Kelly

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New Transmission‐Selective Antimalarial Agents through Hit‐to‐Lead Optimization of 2‐([1,1′‐Biphenyl]‐4‐carboxamido)benzoic Acid Derivatives by Reader, Janette, Opperman, Daniel F. L., Watt, Mariëtte E., Theron, Anjo, Leshabane, Meta, Rocha, Shanté, Turner, Jonathan, Garrabrant, Kathleen, Piña, Ivett, Mills, Catherine, Woster, Patrick M., Birkholtz, Lyn‐Marié

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Potent Plasmodium falciparum gametocytocidal compounds identified by exploring the kinase inhibitor chemical space for dual active antimalarials by van der Watt, Mariëtte E, Reader, Janette, Churchyard, Alisje, Nondaba, Sindisiwe H, Lauterbach, Sonja B, Niemand, Jandeli, Abayomi, Sijuade, van Biljon, Riëtte A, Connacher, Jessica I, van Wyk, Roelof D J, Le Manach, Claire, Paquet, Tanya, González Cabrera, Diego, Brunschwig, Christel, Theron, Anjo, Lozano-Arias, Sonia, Rodrigues, Janneth F I, Herreros, Esperanza, Leroy, Didier, Duffy, James, Street, Leslie J, Chibale, Kelly, Mancama, Dalu, Coetzer, Theresa L, Birkholtz, Lyn-Marie

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The Tuberculosis Drug Candidate SQ109 and Its Analogs Have Multistage Activity against Plasmodium falciparum by Watson, Savannah J., van der Watt, Mariëtte E., Theron, Anjo, Reader, Janette, Tshabalala, Sizwe, Erlank, Erica, Koekemoer, Lizette L., Naude, Mariska, Stampolaki, Marianna, Adewole, Feyisola, Sadowska, Katie, Pérez-Lozano, Pilar, Turcu, Andreea L., Vázquez, Santiago, Ko, Jihee, Mazurek, Ben, Singh, Davinder, Malwal, Satish R., Njoroge, Mathew, Chibale, Kelly, Onajole, Oluseye K., Kolocouris, Antonios, Oldfield, Eric, Birkholtz, Lyn-Marié

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Beskrywing, modellering en dok-studies van Plasmodium falciparum kinase PfCDPK4 by Theron, Anjo, Mancama, Dalu, Van Ree, Teunis, Makungo, Thomas, Tsekoa, Tsepo

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