An Integrated Approach for Identification and Target Validation of Antifungal Compounds Active against Erg11p by HOEPFNER, Dominic, KARKARE, Shantanu, REINKER, Stefan, FREDERIKSEN, Mathias, RAO MOVVA, N, PORTER, Jeffrey A, RYDER, Neil S, PARKER, Christian N, HELLIWELL, Stephen B, PFEIFER, Martin, TRUNZER, Markus, DE BONNECHOSE, Sophie, ZIMMERLIN, Alfred, TAO, Jianshi, RICHIE, Daryl, HOFMANN, Andreas

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Metabolic Soft Spot Identification and Compound Optimization in Early Discovery Phases Using MetaSite and LC-MS/MS Validation by Trunzer, Markus, Faller, Bernard, Zimmerlin, Alfred

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Deep Learning Models Compared to Experimental Variability for the Prediction of CYP3A4 Time-Dependent Inhibition by Fluetsch, Andrin, Trunzer, Markus, Gerebtzoff, Grégori, Rodríguez-Pérez, Raquel

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Multispecies Machine Learning Predictions of In Vitro Intrinsic Clearance with Uncertainty Quantification Analyses by Rodríguez-Pérez, Raquel, Trunzer, Markus, Schneider, Nadine, Faller, Bernard, Gerebtzoff, Grégori

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Design of a Supersoft Topical JAK Inhibitor, Which Is Effective in Human Skin but Rapidly Deactivated in Blood by Thoma, Gebhard, Decoret, Odile, Vangrevelinghe, Eric, Trunzer, Markus, Decker, Andrea, Orjuela Leon, Anette, Beerli, Christian, Bruno, Sandro, Hauchard, Alice, Paulat, Guido, Zerwes, Hans-Guenter, Hacini-Rachinel, Feriel

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Discovery of NP3-253, a Potent Brain Penetrant Inhibitor of the NLRP3 Inflammasome by Mackay, Angela, Velcicky, Juraj, Gommermann, Nina, Mattes, Henri, Janser, Philipp, Wright, Michael, Dubois, Celine, Brenneisen, Silke, Ilic, Slavica, Vangrevelinghe, Eric, Stiefl, Nikolaus, Boettcher, Andreas, Schoenboerner, Michel, Vogelsanger, Melanie, Muller-Bentz, Sophie, Kamke, Marion, Rubert, Joelle, Kauffmann, Muriel, Desrayaud, Sandrine, Trunzer, Markus, Srinivas, Honnappa, Hinniger, Alexandra, von Burg, Nicole, Beltz, Karen, Dekker, Carien, Farady, Christopher J.

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Evaluation of relative MS response factors of drug metabolites for semi‐quantitative assessment of chemical liabilities in drug discovery by Blanz, Joachim, Williams, Gareth, Dayer, Jerôme, Délémonté, Thierry, Gertsch, Werner, Ramstein, Philippe, Aichholz, Reiner, Trunzer, Markus, Pearson, David

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Comparison of a two-dimensional liquid chromatography/mass spectrometry approach with a chip-based nanoelectrospray device for structural elucidation of metabolites in a human ADME... by Trunzer, Markus, Graf, Daniel, Kiffe, Michael

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Two-dimensional liquid chromatography/mass spectrometry set-up for structural elucidation of metabolites in complex biological matrices by Kiffe, Michael, Graf, Daniel, Trunzer, Markus

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Cytostar-T plates—A valid alternative for microplate scintillation counting of low radioactivity in combination with high-performance liquid chromatography in drug metabolism studi... by Kiffe, Michael, Nufer, Robert, Trunzer, Markus, Graf, Daniel

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Photodegradation analysis as additional tool to verify phototoxicity by Struwe, Melanie, Trunzer, Markus, Bauer, Daniel, Kiffe, Michael, Plappert-Helbig, Ulla, Suter, Willi

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System architectures for Industrie 4.0 applications: Derivation of a generic architecture proposal by Trunzer, Emanuel, Calà, Ambra, Leitão, Paulo, Gepp, Michael, Kinghorst, Jakob, Lüder, Arndt, Schauerte, Hubertus, Reifferscheid, Markus, Vogel-Heuser, Birgit

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System architectures for Industrie 4.0 applications by Trunzer, Emanuel, Calà, Ambra, Leitão, Paulo, Gepp, Michael, Kinghorst, Jakob, Arndt Lüder, Schauerte, Hubertus, Reifferscheid, Markus, Vogel-Heuser, Birgit

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