Discovery of Nonpungent Transient Receptor Potential Vanilloid 1 (TRPV1) Agonist as Strong Topical Analgesic by Ann, Jihyae, Kim, Ho Shin, Thorat, Shivaji A, Kim, Hee, Ha, Hee-Jin, Choi, Kwanghyun, Kim, Young-Ho, Kim, Minseok, Hwang, Sun Wook, Pearce, Larry V, Esch, Timothy E, Turcios, Noe A, Blumberg, Peter M, Lee, Jeewoo

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Discovery of Benzopyridone-Based Transient Receptor Potential Vanilloid 1 Agonists and Antagonists and the Structural Elucidation of Their Activity Shift by Thorat, Shivaji A, Lee, Yoonji, Jung, Aeran, Ann, Jihyae, Ahn, Songyeon, Baek, Jisoo, Zuo, Dongxu, Do, Nayeon, Jeong, Jin Ju, Blumberg, Peter M, Esch, Timothy E, Turcios, Noe A, Pearce, Larry V, Ha, Hee-Jin, Yoo, Young Dong, Hong, Sunhye, Choi, Sun, Lee, Jeewoo

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Multi-Functional Diarylurea Small Molecule Inhibitors of TRPV1 with Therapeutic Potential for Neuroinflammation by Feng, Zhiwei, Pearce, Larry V., Zhang, Yu, Xing, Changrui, Herold, Brienna K. A., Ma, Shifan, Hu, Ziheng, Turcios, Noe A., Yang, Peng, Tong, Qin, McCall, Anna K., Blumberg, Peter M., Xie, Xiang-Qun

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Discovery of N-(3-fluoro-4-methylsulfonamidomethylphenyl)urea as a potent TRPV1 antagonistic template by Ann, Jihyae, Sun, Wei, Zhou, Xing, Jung, Aeran, Baek, Jisoo, Lee, Sunho, Kim, Changhoon, Yoon, Suyoung, Hong, Sunhye, Choi, Sun, Turcios, Noe A., Herold, Brienna K.A., Esch, Timothy E., Lewin, Nancy E., Abramovitz, Adelle, Pearce, Larry V., Blumberg, Peter M., Lee, Jeewoo

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2-Sulfonamidopyridine C-region analogs of 2-(3-fluoro-4-methylsulfonamidophenyl)propanamides as potent TRPV1 antagonists by Ann, Jihyae, Ki, Yooran, Yoon, Suyoung, Kim, Myeong Seop, Lee, Jung-Un, Kim, Changhoon, Lee, Sunho, Jung, Aeran, Baek, Jisoo, Hong, Sunhye, Choi, Sun, Pearce, Larry V., Esch, Timothy E., Turcios, Noe A., Lewin, Nancy E., Ogunjirin, Adebowale E., Herold, Brienna K.A., McCall, Anna K., Blumberg, Peter M., Lee, Jeewoo

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