Structure of a small‐molecule inhibitor complexed with GlmU from Haemophilus influenzae reveals an allosteric binding site by Mochalkin, Igor, Lightle, Sandra, Narasimhan, Lakshmi, Bornemeier, Dirk, Melnick, Michael, VanderRoest, Steven, McDowell, Laura

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5,6-Dihydropyran-2-ones Possessing Various Sulfonyl Functionalities:  Potent Nonpeptidic Inhibitors of HIV Protease by Boyer, Frederick E, Vara Prasad, J. V. N, Domagala, John M, Ellsworth, Edmund L, Gajda, Christopher, Hagen, Susan E, Markoski, Larry J, Tait, Bradley D, Lunney, Elizabeth A, Palovsky, Alexander, Ferguson, Donna, Graham, Neil, Holler, Tod, Hupe, Donald, Nouhan, Carolyn, Tummino, Peter J, Urumov, A, Zeikus, Eric, Zeikus, Greg, Gracheck, Stephen J, Sanders, James M, VanderRoest, Steven, Brodfuehrer, Joanne, Iyer, Krishna, Sinz, Michael, Gulnik, Sergei V, Erickson, John W

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Synthesis of 5,6-Dihydro-4-hydroxy-2- pyrones as HIV-1 Protease Inhibitors:  The Profound Effect of Polarity on Antiviral Activity by Hagen, Susan E, Vara Prasad, J. V. N, Boyer, Frederick E, Domagala, John M, Ellsworth, Edmund L, Gajda, Christopher, Hamilton, Harriet W, Markoski, Larry J, Steinbaugh, Bruce A, Tait, Bradley D, Lunney, Elizabeth A, Tummino, Peter J, Ferguson, Donna, Hupe, Donald, Nouhan, Carolyn, Gracheck, Stephen J, Saunders, James M, VanderRoest, Steven

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Comparative therapeutic efficacy of clinafloxacin in leucopenic mice by SHAPIRO, M. A, DEVER, J. A, SESNIE, J. C, VANDERROEST, S. R

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Quinolone antibacterials containing the new 7-[3-(1-aminoethyl)-1-pyrrolidinyl] side chain: the effects of the 1-aminoethyl moiety and its stereochemical configurations on potency... by Domagala, John M, Hagen, Susan E, Joannides, Themis, Kiely, John S, Laborde, Edgardo, Schroeder, Mel C, Sesnie, Josephine A, Shapiro, Martin A, Suto, Mark J, Vanderroest, Steven

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Efficacy of quinolones in preventing Staphylococcus aureus-induced abscess in mice by Cohen, Michael A., Gage, Jeffrey W., Huband, Michael D., Meservey, Mark A., VanderRoest, Steven R., Yoder, Steven L.

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Nonpeptidic HIV protease inhibitors possessing excellent antiviral activities and therapeutic indices. PD 178390 : A lead HIV protease inhibitor by VARA PRASAD, J. V. N, BOYER, F. E, HUMBLET, C, LUNNEY, E. A, PAVLOVSKY, A, RUBIN, J. R, FERGUSON, D, GRAHAM, N, HOLLER, T, HUPE, D, NOUHAN, C, TUMMINO, P. J, DOMAGALA, J. M, URUMOV, A, ZEIKUS, E, ZEIKUS, G, GRACHECK, S. J, SAUNDERS, J. M, VANDERROEST, S, BRODFUEHRER, J, IYER, K, SINZ, M, GULNIK, S. V, ELLSWORTH, E. L, ERICKSON, J. W, GAJDA, C, HAMILTON, H. W, HAGEN, S. E, MARKOSKI, L. J, STEINBAUGH, B. A, TAIT, B. D

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Nonpeptidic HIV protease inhibitors: 6-alkyl-5, 6-dihydropyran-2-ones possessing achiral 3-(4-amino/carboxamide-2- t-butyl, 5-methylphenyl thio) moiety: Antiviral activities and ph... by Vara Prasad, J.V.N., Boyer, Fred E., Domagala, John M., Ellsworth, Edmund L., Gajda, Christopher, Hagen, Susan E., Markoski, Larry J., Tait, Bradley D., Lunney, Elizabeth A., Tummino, Peter J., Ferguson, Donna, Holler, Tod, Hupe, Donald, Nouhan, Carolyn, Gracheck, Stephen J., VanderRoest, Steven, Saunders, James, Iyer, Krishna, Sinz, Michael, Brodfuehrer, Joanne

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Nonpeptidic HIV protease inhibitors: 6-alkyl-5,6-dihydropyran-2-ones possessing a novel and achiral 3-(2- t-butyl-5-methyl-4-sulfamate)phenylthio moiety by Vara Prasad, J.V.N, Markoski, Larry J, Boyer, Fred E, Domagala, John M, Ellsworth, Edmund L, Gajda, Christopher, Hagen, Susan E, Tait, Bradley D, Lunney, Elizabeth A, Tummino, Peter J, Ferguson, Donna, Holler, Tod, Hupe, Donald, Nouhan, Carolyn, Gracheck, Stephen J, VanderRoest, Steven, Saunders, James, Iyer, K, Sinz, M

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