Targeting a Subpocket in Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity by Blaazer, Antoni R, Singh, Abhimanyu K, de Heuvel, Erik, Edink, Ewald, Orrling, Kristina M, Veerman, Johan J. N, van den Bergh, Toine, Jansen, Chimed, Balasubramaniam, Erin, Mooij, Wouter J, Custers, Hans, Sijm, Maarten, Tagoe, Daniel N. A, Kalejaiye, Titilola D, Munday, Jane C, Tenor, Hermann, Matheeussen, An, Wijtmans, Maikel, Siderius, Marco, de Graaf, Chris, Maes, Louis, de Koning, Harry P, Bailey, David S, Sterk, Geert Jan, de Esch, Iwan J. P, Brown, David G, Leurs, Rob

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Discovery of 2,4‑1H‑Imidazole Carboxamides as Potent and Selective TAK1 Inhibitors by Veerman, Johan J. N, Bruseker, Yorik B, Damen, Eddy, Heijne, Erik H, van Bruggen, Wendy, Hekking, Koen F. W, Winkel, Rob, Hupp, Christopher D, Keefe, Anthony D, Liu, Julie, Thomson, Heather A, Zhang, Ying, Cuozzo, John W, McRiner, Andrew J, Mulvihill, Mark J, van Rijnsbergen, Peter, Zech, Birgit, Renzetti, Louis M, Babiss, Lee, Müller, Gerhard

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Synthesis of 2,6-Bridged Piperazine-3-ones by N-Acyliminium Ion Chemistry by Veerman, Johan J. N, Bon, Robin S, Hue, Bui T. B, Girones, Daniel, Rutjes, Floris P. J. T, van Maarseveen, Jan H, Hiemstra, Henk

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Discovery of 2,4-1 H -Imidazole Carboxamides as Potent and Selective TAK1 Inhibitors by Veerman, Johan J N, Bruseker, Yorik B, Damen, Eddy, Heijne, Erik H, van Bruggen, Wendy, Hekking, Koen F W, Winkel, Rob, Hupp, Christopher D, Keefe, Anthony D, Liu, Julie, Thomson, Heather A, Zhang, Ying, Cuozzo, John W, McRiner, Andrew J, Mulvihill, Mark J, van Rijnsbergen, Peter, Zech, Birgit, Renzetti, Louis M, Babiss, Lee, Müller, Gerhard

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Synthesis of Enantiopure Functionalized Pipecolic Acids via Amino Acid Derived N-Acyliminium Ions by Rutjes, Floris P. J. T., Veerman, Johan J. N., Meester, Wim J. N., Hiemstra, Henk, Schoemaker, Hans E.

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Development and application of allyl, 2-sulfonylethyl and 2-thioethyl carbamate linkers for solid phase N-acyliminium ion chemistry by van Maarseveen, Jan H., Meester, Wim J. N., Veerman, Johan J. N., Kruse, Chris G., Hermkens, Pedro H. H., Rutjes, Floris P. J. T., Hiemstra, Henk

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Solid-Phase Synthesis of Piperidines by N-Acyliminium Ion Chemistry by Veerman, Johan J. N., Klein, Jasper, Aben, René W. M., Scheeren, Hans W., Kruse, Chris G., van Maarseveen, Jan H., Rutjes, Floris P. J. T., Hiemstra, Henk

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Synthesis of Enantiopure Functionalized Pipecolic Acids via Amino Acid DerivedN-Acyliminium Ions by Rutjes, Floris P. J. T., Veerman, Johan J. N., Meester, Wim J. N., Hiemstra, Henk, Schoemaker, Hans E.

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Global, regional, and national comparative risk assessment of 84 behavioural, environmental and occupational, and metabolic risks or clusters of risks, 1990–2016: a systematic anal... by Gakidou, Emmanuela, Abate, Kalkidan Hassen, Abd-Allah, Foad, Abdulle, Abdishakur M, Adetokunboh, Olatunji, Agrawal, Sutapa, Al-Aly, Ziyad, Ammar, Walid, Asayesh, Hamid, Azzopardi, Peter, Balakrishnan, Kalpana, Barquera, Simon, Barregard, Lars, Battle, Katherine E, Bennett, James R, Berhe, Derbew Fikadu, Catalá-López, Ferrán, Cercy, Kelly, Dandona, Rakhi, Davletov, Kairat, Dharmaratne, Samath D, Ding, Eric L, Duncan, Bruce Bartholow, El-Khatib, Ziad Ziad, Erskine, Holly E, Esteghamati, Alireza, Farinha, Carla Sofia e Sa, Fullman, Nancy, Furtado, Joao M, Gemechu, Bikila Lencha, Gopalani, Sameer Vali, Handal, Alexis J, Hankey, Graeme J, Horita, Nobuyuki, Jackson, Maria Delores, Johansson, Lars R K, Kahsay, Amaha, Karema, Corine Kakizi, Katikireddi, Srinivasa Vittal, Keiyoro, Peter Njenga, Kiadaliri, Aliasghar Ahmad, Kim, Yun Jin, Kopec, Jacek A, Kyu, Hmwe H, Lalloo, Ratilal, Lee, Paul H, Leigh, James, Li, Yichong, Liu, Patrick, Lopez, Alan D, Lotufo, Paulo A, Lunevicius, Raimundas, Magdy Abd El Razek, Hassan, Mantovani, Lorenzo G, Matzopoulos, Richard, McAlinden, Colm, Mehndiratta, Man Mohan, Melaku, Yohannes Adama, Millear, Anoushka, Mohammed, Kedir Endris, Montico, Marcella, Morawska, Lidia, Musa, Kamarul Imran, Natarajan, Gopalakrishnan, Noubiap, Jean Jacques N, Olagunju, Tinuke Oluwasefunmi, Olusanya, Jacob Olusegun, Panda-Jonas, Songhomitra, Pandian, Jeyaraj D, Papachristou, Christina, Piradov, Michael A, Plass, Dietrich, Pourmalek, Farshad, Reiner, Robert C, Ribeiro, Antonio L, Sadat, Nafis, Safi, Sare, Sanchez-Niño, Maria Dolores, Shaddick, Gavin, Shamsipour, Mansour, Shariful Islam, Sheikh Mohammed, Shen, Jiabin, Shiferaw, Mekonnen Sisay, Smith, David L, Strub, Bryan, Tarekegn, Yihunie L, Tegegne, Teketo Kassaw, Tehrani-Banihashemi, Arash, Thankappan, Kavumpurathu Raman, Thrift, Amanda G, Torre, Anna, Uneke, Chigozie Jesse, Varughese, Santosh, Venkateswaran, Vidhya, Venketasubramanian, Narayanaswamy, Violante, Francesco S, Yakob, Bereket, Yan, Lijing L, Yimam, Hassen Hamid, Zavala-Arciniega, Luis

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