Discovery of First-in-Class PROTAC Degraders of SARS-CoV‑2 Main Protease by Alugubelli, Yugendar R., Xiao, Jing, Khatua, Kaustav, Kumar, Sathish, Sun, Long, Ma, Yuying, Ma, Xinyu R., Vulupala, Veerabhadra R., Atla, Sandeep, Blankenship, Lauren R., Coleman, Demonta, Xie, Xuping, Neuman, Benjamin W., Liu, Wenshe Ray, Xu, Shiqing

Get full text

Azapeptides with unique covalent warheads as SARS-CoV-2 main protease inhibitors by Khatua, Kaustav, Alugubelli, Yugendar R., Yang, Kai S., Vulupala, Veerabhadra R., Blankenship, Lauren R., Coleman, Demonta, Atla, Sandeep, Chaki, Sankar P., Geng, Zhi Zachary, Ma, Xinyu R., Xiao, Jing, Chen, Peng-Hsun, Cho, Chia-Chuan D., Sharma, Shivangi, Vatansever, Erol C., Ma, Yuying, Yu, Ge, Neuman, Benjamin W., Xu, Shiqing, Liu, Wenshe Ray

Get full text

SARS-CoV‑2 Main Protease Inhibitors That Leverage Unique Interactions with the Solvent Exposed S3 Site of the Enzyme by Blankenship, Lauren R., Yang, Kai S., Vulupala, Veerabhadra R., Alugubelli, Yugendar R., Khatua, Kaustav, Coleman, Demonta, Ma, Xinyu R., Sankaran, Banumathi, Cho, Chia-Chuan D., Ma, Yuying, Neuman, Benjamin W., Xu, Shiqing, Liu, Wenshe Ray

Get full text

A Systematic Survey of Reversibly Covalent Dipeptidyl Inhibitors of the SARS-CoV‑2 Main Protease by Geng, Zhi Zachary, Atla, Sandeep, Shaabani, Namir, Vulupala, Veerabhadra, Yang, Kai S., Alugubelli, Yugendar R., Khatua, Kaustav, Chen, Peng-Hsun, Xiao, Jing, Blankenship, Lauren R., Ma, Xinyu R., Vatansever, Erol C., Cho, Chia-Chuan D., Ma, Yuying, Allen, Robert, Ji, Henry, Xu, Shiqing, Liu, Wenshe Ray

Get full text