Structure-Based Design, Synthesis, and Biological Evaluation of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors by Waldschmidt, Helen V, Homan, Kristoff T, Cruz-Rodríguez, Osvaldo, Cato, Marilyn C, Waninger-Saroni, Jessica, Larimore, Kelly M, Cannavo, Alessandro, Song, Jianliang, Cheung, Joseph Y, Kirchhoff, Paul D, Koch, Walter J, Tesmer, John J. G, Larsen, Scott D

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Utilizing a structure-based docking approach to develop potent G protein-coupled receptor kinase (GRK) 2 and 5 inhibitors by Waldschmidt, Helen V., Bouley, Renee, Kirchhoff, Paul D., Lee, Pil, Tesmer, John J.G., Larsen, Scott D.

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Structural Determinants Influencing the Potency and Selectivity of Indazole-Paroxetine Hybrid G Protein–Coupled Receptor Kinase 2 Inhibitors by Bouley, Renee, Waldschmidt, Helen V., Cato, M. Claire, Cannavo, Alessandro, Song, Jianliang, Cheung, Joseph Y., Yao, Xin-Qiu, Koch, Walter J., Larsen, Scott D., Tesmer, John J.G.

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A New Paroxetine-Based GRK2 Inhibitor Reduces Internalization of the μ-Opioid Receptor by Bouley, Renee A., Weinberg, Zara Y., Waldschmidt, Helen V., Yen, Yu-Chen, Larsen, Scott D., Puthenveedu, Manojkumar A., Tesmer, John J.G.

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Small-Molecule G Protein–Coupled Receptor Kinase Inhibitors Attenuate G Protein–Coupled Receptor Kinase 2–Mediated Desensitization of Vasoconstrictor-Induced Arterial Contractions... by Rainbow, Richard D., Brennan, Sean, Jackson, Robert, Beech, Alison J., Bengreed, Amal, Waldschmidt, Helen V., Tesmer, John J.G., Challiss, R.A. John, Willets, Jonathon M.

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Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors Based on Paroxetine by Waldschmidt, Helen V, Homan, Kristoff T, Cato, Marilyn C, Cruz-Rodríguez, Osvaldo, Cannavo, Alessandro, Wilson, Michael W, Song, Jianliang, Cheung, Joseph Y, Koch, Walter J, Tesmer, John J. G, Larsen, Scott D

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Crystal Structure of G Protein-coupled Receptor Kinase 5 in Complex with a Rationally Designed Inhibitor by Homan, Kristoff T., Waldschmidt, Helen V., Glukhova, Alisa, Cannavo, Alessandro, Song, Jianliang, Cheung, Joseph Y., Koch, Walter J., Larsen, Scott D., Tesmer, John J.G.

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Occludin S471 Phosphorylation Contributes to Epithelial Monolayer Maturation by Bolinger, Mark T., Ramshekar, Aniket, Waldschmidt, Helen V., Larsen, Scott D., Bewley, Maria C., Flanagan, John M., Antonetti, David A.

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Correction to “Structure-Based Design of Highly Selective and Potent G Protein-Coupled Receptor Kinase 2 Inhibitors Based on Paroxetine” by Waldschmidt, Helen V, Homan, Kristoff T, Cato, Marilyn C, Cruz-Rodríguez, Osvaldo, Cannavo, Alessandro, Wilson, Michael W, Song, Jianliang, Cheung, Joseph Y, Koch, Walter J, Tesmer, John J. G, Larsen, Scott D

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Structure-Based Design of Selective, Covalent G Protein-Coupled Receptor Kinase 5 Inhibitors by Rowlands, Rachel A, Cato, M. Claire, Waldschmidt, Helen V, Bouley, Renee A, Chen, Qiuyan, Avramova, Larisa, Larsen, Scott D, Tesmer, John J. G, White, Andrew D

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Translation of structure-activity relationships from cyclic mixed efficacy opioid peptides to linear analogues by Anand, Jessica P., Porter-Barrus, Vanessa R., Waldschmidt, Helen V., Yeomans, Larisa, Pogozheva, Irina D., Traynor, John R., Mosberg, Henry I.

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