Development of a new permeability assay using low‐efflux MDCKII cells by Di, Li, Whitney‐Pickett, Carrie, Umland, John P., Zhang, Hui, Zhang, Xun, Gebhard, David F., Lai, Yurong, Federico, James J., Davidson, Ralph E., Smith, Russ, Reyner, Eric L., Lee, Caroline, Feng, Bo, Rotter, Charles, Varma, Manthena V., Kempshall, Sarah, Fenner, Katherine, El‐kattan, Ayman F., Liston, Theodore E., Troutman, Matthew D.

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The JAK-3 inhibitor CP-690550 is a potent anti-inflammatory agent in a murine model of pulmonary eosinophilia by Kudlacz, Elizabeth, Conklyn, Maryrose, Andresen, Catharine, Whitney-Pickett, Carrie, Changelian, Paul

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pH-Dependent Solubility and Permeability Criteria for Provisional Biopharmaceutics Classification (BCS and BDDCS) in Early Drug Discovery by Varma, Manthena V, Gardner, Iain, Steyn, Stefanus J, Nkansah, Paul, Rotter, Charles J, Whitney-Pickett, Carrie, Zhang, Hui, Di, Li, Cram, Michael, Fenner, Katherine S, El-Kattan, Ayman F

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Optimization of the physicochemical and pharmacokinetic attributes in a 6-azauracil series of P2X 7 receptor antagonists leading to the discovery of the clinical candidate CE-224,5... by Duplantier, Allen J., Dombroski, Mark A., Subramanyam, Chakrapani, Beaulieu, Aimee M., Chang, Shang-Poa, Gabel, Christopher A., Jordan, Crystal, Kalgutkar, Amit S., Kraus, Kenneth G., Labasi, Jeff M., Mussari, Christopher, Perregaux, David G., Shepard, Rick, Taylor, Timothy J., Trevena, Kristen A., Whitney-Pickett, Carrie, Yoon, Kwansik

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Discovery, synthesis and SAR of azinyl- and azolylbenzamides antagonists of the P2X7 receptor by Subramanyam, Chakrapani, Duplantier, Allen J., Dombroski, Mark A., Chang, Shang-Poa, Gabel, Christopher A., Whitney-Pickett, Carrie, Perregaux, David G., Labasi, Jeff M., Yoon, Kwansik, Shepard, Richard M., Fisher, Michael

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Synthesis of 12-membered macrocyclic templates and library analogs for PPI by Chen, Jinshan, Rong, Frank, Shan, Bo, Chen, Yuanwei, Li, Yingfu, Yu, Hua, Chen, Li, Kuang, Tongtao, Li, Shai, Chen, Youpei, Du, Jing, Ai, Chaowu, Li, Jian, Li, Xiaoyong, Shi, Changqing, Jiang, Zhilong, Long, Yuanqiang, Gao, Qiu, Wang, Zhibo, Xu, Kexin, Ran, Xin, Yi, Hua, Zhao, Dapeng, Qiao, Hongyun, Shen, Junwei, Liu, Bo, Liu, Chonggang, Wu, Kai, Geng, Xi, Tan, Jieyang, McLeod, Dale, Frost, Heather, Bai, Guoyun, Goetz, Gilles, Federico, James, Whitney-Pickett, Carrie, Troutman, Matthew, Noe, Mark C., Guimaraes, Cristiano, Piotrowski, David W., Magee, Thomas V.

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Discovery, synthesis and SAR of azinyl- and azolylbenzamides antagonists of the P2X sub(7 receptor) by Subramanyam, Chakrapani, Duplantier, Allen J, Dombroski, Mark A, Chang, Shang-Poa, Gabel, Christopher A, Whitney-Pickett, Carrie, Perregaux, David G, Labasi, Jeff M, Yoon, Kwansik, Shepard, Richard M, Fisher, Michael

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Optimization of the physicochemical and pharmacokinetic attributes in a 6-azauracil series of P2X sub(7 receptor antagonists leading to the discovery of the clinical candidate CE-2... by Duplantier, Allen J, Dombroski, Mark A, Subramanyam, Chakrapani, Beaulieu, Aimee M, Chang, Shang-Poa, Gabel, Christopher A, Jordan, Crystal, Kalgutkar, Amit S, Kraus, Kenneth G, Labasi, Jeff M, Mussari, Christopher, Perregaux, David G, Shepard, Rick, Taylor, Timothy J, Trevena, Kristen A, Whitney-Pickett, Carrie, Yoon, Kwansik

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Optimization of the physicochemical and pharmacokinetic attributes in a 6-azauracil series of P2X₇ receptor antagonists leading to the discovery of the clinical candidate CE-224,53... by Duplantier, Allen J, Dombroski, Mark A, Subramanyam, Chakrapani, Beaulieu, Aimee M, Chang, Shang-Poa, Gabel, Christopher A, Jordan, Crystal, Kalgutkar, Amit S, Kraus, Kenneth G, Labasi, Jeff M, Mussari, Christopher, Perregaux, David G, Shepard, Rick, Taylor, Timothy J, Trevena, Kristen A, Whitney-Pickett, Carrie, Yoon, Kwansik

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