The Human Mixed Lineage Leukemia 5 (MLL5), a Sequentially and Structurally Divergent SET Domain-Containing Protein with No Intrinsic Catalytic Activity by Mas-Y-Mas, Sarah, Barbon, Marta, Teyssier, Catherine, Déméné, Hélène, Carvalho, João E, Bird, Louise E, Lebedev, Andrey, Fattori, Juliana, Schubert, Michael, Dumas, Christian, Bourguet, William, le Maire, Albane

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A Comparative Study of Human and Zebrafish Pregnane X Receptor Activities of Pesticides and Steroids Using In Vitro Reporter Gene Assays by Creusot, Nicolas, Garoche, Clémentine, Grimaldi, Marina, Boulahtouf, Abdelhay, Chiavarina, Barbara, Bourguet, William, Balaguer, Patrick

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What Structural Biology Tells Us About the Mode of Action and Detection of Toxicants by le Maire, Albane, Bourguet, William

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An Unexpected Mode Of Binding Defines BMS948 as A Full Retinoic Acid Receptor β (RARβ, NR1B2) Selective Agonist by Nadendla, Eswarkumar, Teyssier, Catherine, Delfosse, Vanessa, Vivat, Valérie, Krishnasamy, Gunasekaran, Gronemeyer, Hinrich, Bourguet, William, Germain, Pierre

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A Mollusk Retinoic Acid Receptor (RAR) Ortholog Sheds Light on the Evolution of Ligand Binding by Gutierrez-Mazariegos, Juliana, Nadendla, Eswar Kumar, Lima, Daniela, Pierzchalski, Keely, Jones, Jace W, Kane, Maureen, Nishikawa, Jun-Ichi, Hiromori, Youhei, Nakanishi, Tsuyoshi, Santos, Miguel M, Castro, L. Filipe C, Bourguet, William, Schubert, Michael, Laudet, Vincent

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Modulators of the structural dynamics of the retinoid X receptor to reveal receptor function by Nahoum, Virginie, Pérez, Efrén, Germain, Pierre, Rodríguez-Barrios, Fátima, Manzo, Fabio, Kammerer, Sabrina, Lemaire, Geraldine, Hirsch, Oliver, Royer, Catherine A, Gronemeyer, Hinrich, de Lera, Angel R, Bourguet, William

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Structural and Functional Evidence for Ligand-Independent Transcriptional Activation by the Estrogen-Related Receptor 3 by Greschik, Holger, Wurtz, Jean-Marie, Sanglier, Sarah, Bourguet, William, van Dorsselaer, Alain, Moras, Dino, Renaud, Jean-Paul

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High Content Screening Using New U2OS Reporter Cell Models Identifies Harmol Hydrochloride as a Selective and Competitive Antagonist of the Androgen Receptor by Dellal, Hadjer, Boulahtouf, Abdelhay, Alaterre, Elina, Cuenant, Alice, Grimaldi, Marina, Bourguet, William, Gongora, Céline, Balaguer, Patrick, Pourquier, Philippe

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Development of new approach methods for the identification and characterization of endocrine metabolic disruptors-a PARC project by Braeuning, Albert, Balaguer, Patrick, Bourguet, William, Carreras-Puigvert, Jordi, Feiertag, Katreece, Kamstra, Jorke H, Knapen, Dries, Lichtenstein, Dajana, Marx-Stoelting, Philip, Rietdijk, Jonne, Schubert, Kristin, Spjuth, Ola, Stinckens, Evelyn, Thedieck, Kathrin, van den Boom, Rik, Vergauwen, Lucia, von Bergen, Martin, Wewer, Neele, Zalko, Daniel

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Crystal Structure of a Heterodimeric Complex of RAR and RXR Ligand-Binding Domains by Bourguet, William, Vivat, Valérie, Wurtz, Jean-Marie, Chambon, Pierre, Gronemeyer, Hinrich, Moras, Dino

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Corrigendum: Development of new approach methods for the identification and characterization of endocrine metabolic disruptors-a PARC project by Braeuning, Albert, Balaguer, Patrick, Bourguet, William, Carreras-Puigvert, Jordi, Feiertag, Katreece, Kamstra, Jorke H, Knapen, Dries, Lichtenstein, Dajana, Marx-Stoelting, Philip, Rietdijk, Jonne, Schubert, Kristin, Spjuth, Ola, Stinckens, Evelyn, Thedieck, Kathrin, van den Boom, Rik, Vergauwen, Lucia, von Bergen, Martin, Wewer, Neele, Zalko, Daniel

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The ancestral retinoic acid receptor was a low-affinity sensor triggering neuronal differentiation by Handberg-Thorsager, Mette, Gutierrez-Mazariegos, Juliana, Arold, Stefan T, Kumar Nadendla, Eswar, Bertucci, Paola Y, Germain, Pierre, Tomançak, Pavel, Pierzchalski, Keely, Jones, Jace W, Albalat, Ricard, Kane, Maureen A, Bourguet, William, Laudet, Vincent, Arendt, Detlev, Schubert, Michael

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Characterization of the Interaction between Retinoic Acid Receptor/Retinoid X Receptor (RAR/RXR) Heterodimers and Transcriptional Coactivators through Structural and Fluorescence A... by Pogenberg, Vivian, Guichou, Jean-François, Vivat-Hannah, Valérie, Kammerer, Sabrina, Pérez, Efrén, Germain, Pierre, de Lera, Angel R., Gronemeyer, Hinrich, Royer, Catherine A., Bourguet, William

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Evolutionary diversification of retinoic acid receptor ligand-binding pocket structure by molecular tinkering by Gutierrez-Mazariegos, Juliana, Nadendla, Eswar Kumar, Studer, Romain A., Alvarez, Susana, de Lera, Angel R., Kuraku, Shigehiro, Bourguet, William, Schubert, Michael, Laudet, Vincent

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In Silico Predictions of Endocrine Disruptors Properties by Schneider, Melanie, Pons, Jean-Luc, Labesse, Gilles, Bourguet, William

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Towards accurate high-throughput ligand affinity prediction by exploiting structural ensembles, docking metrics and ligand similarity by Schneider, Melanie, Pons, Jean-Luc, Bourguet, William, Labesse, Gilles

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Separation of Retinoid X Receptor Homo- and Heterodimerization Functions by Vivat-Hannah, Valerie, Bourguet, William, Gottardis, Marco, Gronemeyer, Hinrich

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Mechanistic insights into the synergistic activation of the RXR–PXR heterodimer by endocrine disruptor mixtures by Delfosse, Vanessa, Huet, Tiphaine, Harrus, Deborah, Granell, Meritxell, Bourguet, Maxime, Gardia-Parège, Caroline, Chiavarina, Barbara, Grimaldi, Marina, Le Mével, Sébastien, Blanc, Pauline, Huang, David, Gruszczyk, Jakub, Demeneix, Barbara, Cianférani, Sarah, Fini, Jean-Baptiste, Balaguer, Patrick, Bourguet, William

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Interspecies Differences in Activation of Peroxisome Proliferator-Activated Receptor γ by Pharmaceutical and Environmental Chemicals by Garoche, Clémentine, Boulahtouf, Abdelhay, Grimaldi, Marina, Chiavarina, Barbara, Toporova, Lucia, den Broeder, Marjo J, Legler, Juliette, Bourguet, William, Balaguer, Patrick

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Peroxisome Proliferator-Activated Receptor γ Is a Target for Halogenated Analogs of Bisphenol A by Riu, Anne, Grimaldi, Marina, le Maire, Albane, Bey, Gilbert, Phillips, Kevin, Boulahtouf, Abdelhay, Perdu, Elisabeth, Zalko, Daniel, Bourguet, William, Balaguer, Patrick

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