Pharmacological and immunohistochemical characterization of the APJ receptor and its endogenous ligand apelin by Medhurst, Andrew D., Jennings, Carol A., Robbins, Melanie J., Davis, Robert P., Ellis, Catherine, Winborn, Kim Y., Lawrie, Kenneth W. M., Hervieu, Guillaume, Riley, Graham, Bolaky, Jane E., Herrity, Nicole C., Murdock, Paul, Darker, John G.

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Design and Synthesis of trans-3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))- phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro- 1H-3-benzazepine (SB-414796): ... by Macdonald, Gregor J, Branch, Clive L, Hadley, Michael S, Johnson, Christopher N, Nash, David J, Smith, Alexander B, Stemp, Geoffrey, Thewlis, Kevin M, Vong, Antonio K. K, Austin, Nigel E, Jeffrey, Phillip, Winborn, Kim Y, Boyfield, Izzy, Hagan, Jim J, Middlemiss, Derek N, Reavill, Charlie, Riley, Graham J, Watson, Jeannette M, Wood, Martyn, Parker, Steve G, Ashby, Charles R

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Design and synthesis of 6-phenylnicotinamide derivatives as antagonists of TRPV1 by Westaway, Susan M., Thompson, Mervyn, Rami, Harshad K., Stemp, Geoffrey, Trouw, Leontine S., Mitchell, Darren J., Seal, Jon T., Medhurst, Stephen J., Lappin, Sarah C., Biggs, James, Wright, James, Arpino, Sandra, Jerman, Jeffrey C., Cryan, Jennifer E., Holland, Vicky, Winborn, Kim Y., Coleman, Tanya, Stevens, Alexander J., Davis, John B., Gunthorpe, Martin J.

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SAR of biphenyl carboxamide ligands of the human melanin-concentrating hormone receptor 1 (MCH R1): Discovery of antagonist SB-568849 by Witty, David R., Bateson, John H., Hervieu, Guillaume J., Jeffrey, Phillip, Johnson, Christopher N., Muir, Alison I., O’Hanlon, Peter J., Stemp, Geoffrey, Stevens, Alex J., Thewlis, Kevin M., Wilson, Shelagh, Winborn, Kim Y.

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Discovery of potent and stable conformationally constrained analogues of the MCH R1 antagonist SB-568849 by Witty, David R., Bateson, John, Hervieu, Guillaume J., Al-Barazanji, Kamal, Jeffrey, Phillip, Hamprecht, Dieter, Haynes, Andrea, Johnson, Christopher N., Muir, Alison I., O’Hanlon, Peter J., Stemp, Geoffrey, Stevens, Alex J., Thewlis, Kevin, Winborn, Kim Y.

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N-Tetrahydroquinolinyl, N-quinolinyl and N-isoquinolinyl biaryl carboxamides as antagonists of TRPV1 by Westaway, Susan M., Chung, Ying-Kit, Davis, John B., Holland, Vicky, Jerman, Jeffrey C., Medhurst, Stephen J., Rami, Harshad K., Stemp, Geoffrey, Stevens, Alexander J., Thompson, Mervyn, Winborn, Kim Y., Wright, James

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Design and Synthesis of trans -3-(2-(4-((3-(3-(5-Methyl-1,2,4-oxadiazolyl))- phenyl)carboxamido)cyclohexyl)ethyl)-7-methylsulfonyl-2,3,4,5-tetrahydro- 1 H -3-benzazepine (SB-414796... by Macdonald, Gregor J., Branch, Clive L., Hadley, Michael S., Johnson, Christopher N., Nash, David J., Smith, Alexander B., Stemp, Geoffrey, Thewlis, Kevin M., Vong, Antonio K. K., Austin, Nigel E., Jeffrey, Phillip, Winborn, Kim Y., Boyfield, Izzy, Hagan, Jim J., Middlemiss, Derek N., Reavill, Charlie, Riley, Graham J., Watson, Jeannette M., Wood, Martyn, Parker, Steve G., Ashby, Charles R.

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Design and synthesis of trans-3-2-4-3-(3-(5-methyl-1,2,4-oxadiazolyl))-phenylcarboxamidocyclohexyl ethyl-7-methylsulfonyl-2,3,4,5-tetrahydro-1H-3-benzazepine (SB-414796): A potent... by MACDONALD, Gregor J, BRANCH, Clive L, JEFFREY, Phillip, WINBORN, Kim Y, BOYFIELD, Izzy, HAGAN, Jim J, MIDDLEMISS, Derek N, REAVILL, Charlie, RILEY, Graham J, WATSON, Jeannette M, WOOD, Martyn, PARKER, Steve G, HADLEY, Michael S, ASHBY, Charles R, JOHNSON, Christopher N, NASH, David J, SMITH, Alexander B, STEMP, Geoffrey, THEWLIS, Kevin M, VONG, Antonio K. K, AUSTIN, Nigel E

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