Discovery of β‑Arrestin Biased, Orally Bioavailable, and CNS Penetrant Neurotensin Receptor 1 (NTR1) Allosteric Modulators by Pinkerton, Anthony B, Peddibhotla, Satyamaheshwar, Yamamoto, Fusayo, Slosky, Lauren M, Bai, Yushi, Maloney, Patrick, Hershberger, Paul, Hedrick, Michael P, Falter, Bekhi, Ardecky, Robert J, Smith, Layton H, Chung, Thomas D. Y, Jackson, Michael R, Caron, Marc G, Barak, Lawrence S

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(1S)-1,5-Anhydro-1-[5-(4-ethoxybenzyl)-2-methoxy-4-methylphenyl]-1-thio-d-glucitol (TS-071) is a Potent, Selective Sodium-Dependent Glucose Cotransporter 2 (SGLT2) Inhibitor for Ty... by Kakinuma, Hiroyuki, Oi, Takahiro, Hashimoto-Tsuchiya, Yuko, Arai, Masayuki, Kawakita, Yasunori, Fukasawa, Yoshiki, Iida, Izumi, Hagima, Naoko, Takeuchi, Hiroyuki, Chino, Yukihiro, Asami, Jun, Okumura-Kitajima, Lisa, Io, Fusayo, Yamamoto, Daisuke, Miyata, Noriyuki, Takahashi, Teisuke, Uchida, Saeko, Yamamoto, Koji

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Discovery of potent, low-absorbable sodium-dependent glucose cotransporter 1 (SGLT1) inhibitor SGL5213 for type 2 diabetes treatment by Kuroda, Shoichi, Kobashi, Yohei, Oi, Takahiro, Kawabe, Kenichi, Shiozawa, Fumiyasu, Okumura-Kitajima, Lisa, Sugisaki-Kitano, Mami, Io, Fusayo, Yamamoto, Koji, Kakinuma, Hiroyuki

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TP0463518, a Novel Prolyl Hydroxylase Inhibitor, Specifically Induces Erythropoietin Production in the Liver by Kato, Sota, Ochiai, Nagahiro, Takano, Hiroki, Io, Fusayo, Takayama, Noriko, Koretsune, Hiroko, Kunioka, Ei-ichi, Uchida, Saeko, Yamamoto, Koji

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Lenvatinib, an angiogenesis inhibitor targeting VEGFR/FGFR, shows broad antitumor activity in human tumor xenograft models associated with microvessel density and pericyte coverage by Yamamoto, Yuji, Matsui, Junji, Matsushima, Tomohiro, Obaishi, Hiroshi, Miyazaki, Kazuki, Nakamura, Katsuji, Tohyama, Osamu, Semba, Taro, Yamaguchi, Atsumi, Hoshi, Sachi Suzuki, Mimura, Fusayo, Haneda, Toru, Fukuda, Yoshio, Kamata, Jun-Ichi, Takahashi, Keiko, Matsukura, Masayuki, Wakabayashi, Toshiaki, Asada, Makoto, Nomoto, Ken-Ichi, Watanabe, Tatsuo, Dezso, Zoltan, Yoshimatsu, Kentaro, Funahashi, Yasuhiro, Tsuruoka, Akihiko

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Immunoreactivity of TTF‐1, GATA‐3, CEA, and p16/Ki67 cocktail in Cellprep®‐processed control samples: Comparison of long‐term storage in vials and slides by Ryu, Ayumi, Honma, Keiichiro, Umeno, Yoshimi, Uefuji, Fusayo, Muramatsu, Takako, Nishimura, Sanako, Tanada, Satoshi, Yamamoto, Takashi, Nagata, Shigenori, Yamasaki, Tomoyuki, Ohue, Masayuki

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Real-World Methotrexate Dose on Clinical Effectiveness and Structural Damage of Certolizumab Pegol With Rheumatoid Arthritis by Nozaki, Yuji, Hidaka, Toshihiko, Ri, Jinhai, Itami, Tetsu, Tomita, Daisuke, Okada, Akinori, Ashida, Chisato, Ikeda, Fusayo, Yamamoto, Atsuhiro, Funahashi, Keiko, Kinoshita, Koji, Matsubara, Tsukasa, Funauchi, Masanori, Matsumura, Itaru

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Discovery of novel (4-piperidinyl)-piperazines as potent and orally active acetyl-CoA carboxylase 1/2 non-selective inhibitors: F-Boc and triF-Boc groups are acid-stable bioisoster... by Chonan, Tomomichi, Wakasugi, Daisuke, Yamamoto, Daisuke, Yashiro, Miyoko, Oi, Takahiro, Tanaka, Hiroaki, Ohoka-Sugita, Ayumi, Io, Fusayo, Koretsune, Hiroko, Hiratate, Akira

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SGL5213, a novel and potent intestinal SGLT1 inhibitor, suppresses intestinal glucose absorption and enhances plasma GLP-1 and GLP-2 secretion in rats by Io, Fusayo, Gunji, Emi, Koretsune, Hiroko, Kato, Koji, Sugisaki-Kitano, Mami, Okumura-Kitajima, Lisa, Kimura, Kayo, Uchida, Saeko, Yamamoto, Koji

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Design and synthesis of disubstituted (4-piperidinyl)-piperazine derivatives as potent acetyl-CoA carboxylase inhibitors by Chonan, Tomomichi, Tanaka, Hiroaki, Yamamoto, Daisuke, Yashiro, Miyoko, Oi, Takahiro, Wakasugi, Daisuke, Ohoka-Sugita, Ayumi, Io, Fusayo, Koretsune, Hiroko, Hiratate, Akira

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(4-Piperidinyl)-piperazine: A new platform for acetyl-CoA carboxylase inhibitors by Chonan, Tomomichi, Oi, Takahiro, Yamamoto, Daisuke, Yashiro, Miyoko, Wakasugi, Daisuke, Tanaka, Hiroaki, Ohoka-Sugita, Ayumi, Io, Fusayo, Koretsune, Hiroko, Hiratate, Akira

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