Quinol-4-ones as Steroid A-Ring Mimetics in Nonsteroidal Dissociated Glucocorticoid Agonists by Regan, John, Lee, Thomas W, Zindell, Renée M, Bekkali, Younes, Bentzien, Jörg, Gilmore, Thomas, Hammach, Abdelhakim, Kirrane, Thomas M, Kukulka, Alison J, Kuzmich, Daniel, Nelson, Richard M, Proudfoot, John R, Ralph, Mark, Pelletier, Josephine, Souza, Donald, Zuvela-Jelaska, Lijiljana, Nabozny, Gerald, Thomson, David S

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Trifluoromethyl group as a pharmacophore : Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand by BETAGERI, Raj, YAN ZHANG, PAW, Zofia, SHIH, Daw-Tsun, SHIH, Cheng-Kon, ZUVELA-JELASKA, Ljiljana, NABOZNY, Gerald, THOMSON, David S, ZINDELL, Renee M, KUZMICH, Daniel, KIRRANE, Thomas M, BENTZIEN, Jörg, CARDOZO, Mario, CAPOLINO, Alison J, FADRA, Tazmeen N, NELSON, Richard M

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Synthesis, SAR, and Series Evolution of Novel Oxadiazole-Containing 5‑Lipoxygenase Activating Protein Inhibitors: Discovery of 2‑[4-(3-{(R)‑1-[4-(2-Amino-pyrimidin-5-yl)-phenyl]-1-... by Takahashi, Hidenori, Riether, Doris, Bartolozzi, Alessandra, Bosanac, Todd, Berger, Valentina, Binetti, Ralph, Broadwater, John, Chen, Zhidong, Crux, Rebecca, De Lombaert, Stéphane, Dave, Rajvee, Dines, Jonathon A, Fadra-Khan, Tazmeen, Flegg, Adam, Garrigou, Michael, Hao, Ming-Hong, Huber, John, Hutzler, J. Matthew, Kerr, Steven, Kotey, Adrian, Liu, Weimin, Lo, Ho Yin, Loke, Pui Leng, Mahaney, Paige E, Morwick, Tina M, Napier, Spencer, Olague, Alan, Pack, Edward, Padyana, Anil K, Thomson, David S, Tye, Heather, Wu, Lifen, Zindell, Renee M, Abeywardane, Asitha, Simpson, Thomas

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Discovery and optimization of oxadiazole-based FLAP inhibitors by Bartolozzi, Alessandra, Abeywardane, Asitha, Bosanac, Todd, Broadwater, John A., Chen, Zhidong, Hutzler, J. Matthew, Huber, John D., Nemoto, Peter, Olague, Alan, Riether, Doris, Simpson, Tom, Takahashi, Hidenori, Wu, Lifen, Zhang, Yunlong, Zindell, Renee M.

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Trifluoromethyl group as a pharmacophore: Effect of replacing a CF 3 group on binding and agonist activity of a glucocorticoid receptor ligand by Betageri, Raj, Zhang, Yan, Zindell, Renee M., Kuzmich, Daniel, Kirrane, Thomas M., Bentzien, Jörg, Cardozo, Mario, Capolino, Alison J., Fadra, Tazmeen N., Nelson, Richard M., Paw, Zofia, Shih, Daw-Tsun, Shih, Cheng-Kon, Zuvela-Jelaska, Ljiljana, Nabozny, Gerald, Thomson, David S.

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Binding Site Elucidation of Hydantoin-Based Antagonists of LFA-1 Using Multidisciplinary Technologies:  Evidence for the Allosteric Inhibition of a Protein−Protein Interaction by Last-Barney, Kathleen, Davidson, Walter, Cardozo, Mario, Frye, Leah L, Grygon, Christine A, Hopkins, Jerry L, Jeanfavre, Deborah D, Pav, Susan, Qian, Chungeng, Stevenson, James M, Tong, Liang, Zindell, Renee, Kelly, Terence A

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Selective CB2 receptor agonists. Part 2: Structure–activity relationship studies and optimization of proline-based compounds by Riether, Doris, Zindell, Renee, Wu, Lifen, Betageri, Raj, Jenkins, James E., Khor, Someina, Berry, Angela K., Hickey, Eugene R., Ermann, Monika, Albrecht, Claudia, Ceci, Angelo, Gemkow, Mark J., Nagaraja, Nelamangala V., Romig, Helmut, Sauer, Achim, Thomson, David S.

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5-Aminomethylbenzimidazoles as potent ITK antagonists by RIETHER, Doris, ZINDELL, Renée, RAYMOND, Ernest L, KHINE, Hnin Hnin, O'SHEA, Kathy, WOSKA, Joseph R, JEANFAVRE, Deborah, SELLATI, Rosemarie, RALPH, Kerry L. M, AHLBERG, Jennifer, LABISSIERE, Gabriel, KASHEM, Mohammed A, KOWALSKI, Jennifer A, PULLEN, Steven S, TAKAHASHI, Hidenori, COOK, Brian N, BENTZIEN, Jörg, DE LOMBAERT, Stéphane, THOMSON, David, KUGLER, Stanley Z, SKOW, Donna, MARTIN, Leslie S

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Design and Synthesis of Dipeptide Nitriles as Reversible and Potent Cathepsin S Inhibitors by Ward, Yancey D, Thomson, David S, Frye, Leah L, Cywin, Charles L, Morwick, Tina, Emmanuel, Michel J, Zindell, Renée, McNeil, Daniel, Bekkali, Younes, Hrapchak, Matt, DeTuri, Molly, Crane, Kathy, White, Della, Pav, Susan, Wang, Yong, Hao, Ming-Hong, Grygon, Christine A, Labadia, Mark E, Freeman, Dorothy M, Davidson, Walter, Hopkins, Jerry L, Brown, Maryanne L, Spero, Denice M

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Design and Synthesis of Dipeptide Nitriles as Reversible and Potent Cathepsin S Inhibitors by Ward, Yancey D, Thomson, David S, Frye, Leah L, Cywin, Charles L, Morwick, Tina, Emmanuel, Michel J, Zindell, Renée, McNeil, Daniel, Bekkali, Younes, Girardot, Marc, Hrapchak, Matt, DeTuri, Molly, Crane, Kathy, White, Della, Pav, Susan, Wang, Yong, Hao, Ming-Hong, Grygon, Christine A, Labadia, Mark E, Freeman, Dorothy M, Davidson, Walter, Hopkins, Jerry L, Brown, Maryanne L, Spero, Denice M

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