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Exploring the SAR of the β‑Ketoacyl-ACP Synthase Inhibitor GSK3011724A and Optimization around a Genotoxic Metabolite by Cunningham, Fraser, Esquivias, Jorge, Fernández-Menéndez, Raquel, Pérez, Arancha, Guardia, Ana, Escribano, Jaime, Rivero, Cristina, Vimal, Mythily, Cacho, Mónica, de Dios-Antón, Paco, Martínez-Martínez, María Santos, Jiménez, Elena, Huertas Valentín, Leticia, Rebollo-López, María José, López-Román, Eva María, Sousa-Morcuende, Verónica, Rullas, Joaquín, Neu, Margaret, Chung, Chun-wa, Bates, Robert H

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Mycobacterium tuberculosis Decaprenylphosphoryl-β‑d‑ribose Oxidase Inhibitors: Expeditious Reconstruction of Suboptimal Hits into a Series with Potent in Vivo Activity by Borthwick, Jennifer A, Alemparte, Carlos, Wall, Ian, Whitehurst, Benjamin C, Argyrou, Argyrides, Burley, Glenn, de Dios-Anton, Paco, Guijarro, Laura, Monteiro, Maria Candida, Ortega, Fatima, Suckling, Colin J, Pichel, Julia Castro, Cacho, Monica, Young, Robert J

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