Structure-Activity Studies on the Corticotropin Releasing Factor Antagonist Astressin, leading to a Minimal Sequence necessary for Antagonistic Activity by Rijkers, Dirk T.S, Kruijtzer, John A.W, van Oostenbrugge, Marja, Ronken, Eric, den Hartog, Jack A.J, Liskamp, Rob M.J

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Solid-phase synthesis of peptidosulfonamide containing peptides derived from Leu-enkephalin by de Bont, Dries B.A, Dijkstra, Gerard D.H, den Hartog, Jack A.J, Liskamp, Rob M.J

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A straightforward synthesis of 1,3-dichloro-5,8-dihydroisoquinoline by consecutive Stille cross-coupling and metathesis reactions by van den Hoogenband, Adri, den Hartog, Jack A.J., Faber-Hilhorst, Nancy, Lange, Jos H.M., Terpstra, Jan Willem

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An efficient synthesis of 4-bromo-N-substituted oxindoles by an intramolecular copper-catalyzed amidation reaction by van den Hoogenband, Adri, Lange, Jos H.M., den Hartog, Jack A.J., Henzen, Remco, Terpstra, Jan Willem

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Design and Synthesis of an orally active GPIIb/IIIa antagonist based on a phenylpiperazine scaffold by van Maarseveen, Jan H, den Hartog, Jack A.J, Tipker, Koos, Reinders, Jan-Hendrik, Brakkee, Joost, Schön, Uwe, Kehrbach, Wolfgang, Kruse, Chris G

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An efficient one-pot synthesis of novel 4-aryl-1-methyloxindoles by van den Hoogenband, Adri, Lange, Jos H.M., Iwema-Bakker, Wouter I., den Hartog, Jack A.J., van Schaik, Jord, Feenstra, Rolf W., Terpstra, Jan Willem

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A novel synthesis of N-(piperidin-4-yl)-1,3-dihydroindol-2-one via an intramolecular Pd-catalyzed amination by van den Hoogenband, Adri, den Hartog, Jack A.J., Lange, Jos H.M., Terpstra, Jan Willem

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Solid phase ring-closing metathesis: Cyclization/cleavage approach towards a seven membered cycloolefin by van Maarseveen, Jan H., den Hartog, Jack A.J., Engelen, Victor, Finner, Emil, Visser, Geb, Kruse, Chris G.

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Synthesis and biological activity of N-terminal lipidated and/or fluorescently labeled conjugates of astressin as corticotropin releasing factor antagonists by Rijkers, Dirk T.S., den Hartog, Jack A.J., Liskamp, Rob M.J.

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An optimized solid phase synthesis strategy- including on-resin lactamization-of astressin, its retro-, inverso-, and retro-inverso isomers as corticotropin releasing factor antago... by Rijkers, Dirk T. S., den Hartog, Jack A. J., Liskamp, Rob M. J.

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Two novel syntheses of the histamine H3 antagonist thioperamide by Lange, Jos H.M., Wals, Henri C., den Hoogenband, Adri van, de Kuilen, Aalt van, den Hartog, Jack A.J.

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Chemical synthesis of a messenger ribonucleic acid fragment: AUGUUCUUCUUCUUCUUC by den Hartog, J A, Wille, G, Scheublin, R A, van Boom, J H

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