Synthesis and characterization of new biologically active 2-(1,3-disubstituted pyrazolyl)chromones and corresponding pyrimidine, thiopyrimidine, pyrazolyl derivatives

A series of 2‐(1‐methyl‐3‐n‐propylpyrazol‐5‐yl)‐chromones with interesting Phosphodiesterase IV inhibitition activities were synthesized. Different derivatives of the titled compounds like aminopyrimidine, thiopyrimidine, pyrazolyl were synthesized and their Phosphodiesterase IV inhibitition activit...

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Published in:Journal of heterocyclic chemistry 2004-07, Vol.41 (4), p.541-548
Main Authors: Joshia, N. S., Karale, B. K., Gill, C. H., Bhirud, S. B.
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Language:English
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cited_by cdi_FETCH-LOGICAL-c3290-a39248ec1a0ac592bc4aae708e29f5abd63de5739140b93d5e1f10d329fb047a3
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container_end_page 548
container_issue 4
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container_title Journal of heterocyclic chemistry
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creator Joshia, N. S.
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description A series of 2‐(1‐methyl‐3‐n‐propylpyrazol‐5‐yl)‐chromones with interesting Phosphodiesterase IV inhibitition activities were synthesized. Different derivatives of the titled compounds like aminopyrimidine, thiopyrimidine, pyrazolyl were synthesized and their Phosphodiesterase IV inhibitition activities were checked.
doi_str_mv 10.1002/jhet.5570410410
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title Synthesis and characterization of new biologically active 2-(1,3-disubstituted pyrazolyl)chromones and corresponding pyrimidine, thiopyrimidine, pyrazolyl derivatives
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