Convenient synthesis of [3R-(3α,4β,5α,6β)]-2-[7-chloro-1-(4-ethylbenzyl)-5-methyl-1H-indol-3-yl]-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol

A novel and convenient approach for the preparation of [3 R -(3α,4β,5α,6β)]-2-[7-chloro-1-(4-ethylbenzyl)-5-methyl-1 H -indol-3-yl]-6-(hydroxymethyl)tetrahydro-2 H -pyran-3,4,5-triol is developed. It has been achieved in about 72% overall yield. Graphical abstract

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Bibliographic Details
Published in:Monatshefte für Chemie 2010-08, Vol.141 (8), p.913-916
Main Authors: Liu, Yong-Hai, Li, Da-Li, Li, Qin-Hua, Yang, Jun-Fang, Lu, Lu-De
Format: Article
Language:English
Subjects:
Analytical Chemistry
Chemistry
Chemistry and Materials Science
Chemistry/Food Science
Inorganic Chemistry
Organic Chemistry
Original Paper
Physical Chemistry
Theoretical and Computational Chemistry
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Summary:A novel and convenient approach for the preparation of [3 R -(3α,4β,5α,6β)]-2-[7-chloro-1-(4-ethylbenzyl)-5-methyl-1 H -indol-3-yl]-6-(hydroxymethyl)tetrahydro-2 H -pyran-3,4,5-triol is developed. It has been achieved in about 72% overall yield. Graphical abstract
ISSN:0026-9247
1434-4475
DOI:10.1007/s00706-010-0350-0