Intramolecular Heck reaction of 2- and 3-iodoindole derivatives for the synthesis of β- and γ-carbolinones

A new synthesis of β- and γ-carbolinone derivatives was achieved by an intramolecular Heck cyclisation from the corresponding 3-iodo-1 H-indole-2-carboxylic acid allyl-amides 8 and 2-iodo-1 H-indole-3-carboxylic acid allyl-amides 9 . Graphic

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Bibliographic Details
Published in:Tetrahedron 2002-08, Vol.58 (33), p.6673-6678
Main Authors: Beccalli, Egle M, Broggini, Gianluigi, Marchesini, Alessandro, Rossi, Elisabetta
Format: Article
Language:English
Subjects:
carbolines
Heck reaction
indoles
intramolecular cyclization
Pd catalyst
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Summary:A new synthesis of β- and γ-carbolinone derivatives was achieved by an intramolecular Heck cyclisation from the corresponding 3-iodo-1 H-indole-2-carboxylic acid allyl-amides 8 and 2-iodo-1 H-indole-3-carboxylic acid allyl-amides 9 . Graphic
ISSN:0040-4020
1464-5416
DOI:10.1016/S0040-4020(02)00688-9