Synthesis of 3-Phenylindoline-2-carboxamides as Semi-Rigid Phenylalanine Mimetics

Regioselective catalytic hydrogenation of N-acyl 3-phenylindole-2-carboxylates is the key step for the preparation of cis and trans indoline-2-carboxamides which can be considered as phenylalanine semi-rigid derivatives. © 1997 Published by Elsevier Science Ltd.

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Bibliographic Details
Published in:Tetrahedron letters 1997-11, Vol.38 (46), p.8033-8036
Main Authors: Collot, Valérie, Schmitt, Martine, Marwah, Ashok K, Norberg, Bernadette, Bourguignon, Jean-Jacques
Format: Article
Language:English
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Summary:Regioselective catalytic hydrogenation of N-acyl 3-phenylindole-2-carboxylates is the key step for the preparation of cis and trans indoline-2-carboxamides which can be considered as phenylalanine semi-rigid derivatives. © 1997 Published by Elsevier Science Ltd.
ISSN:0040-4039
1873-3581
DOI:10.1016/S0040-4039(97)10214-3