Structure-Based Design and Synthesis of 3-Amino-1,5-dihydro-4 H -pyrazolopyridin-4-one Derivatives as Tyrosine Kinase 2 Inhibitors

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Published in:Journal of medicinal chemistry 2016-01, Vol.59 (2), p.733-749
Main Authors: Yogo, Takatoshi, Nagamiya, Hiroyuki, Seto, Masaki, Sasaki, Satoshi, Shih-Chung, Huang, Ohba, Yusuke, Tokunaga, Norihito, Lee, Gil Nam, Rhim, Chul Yun, Yoon, Cheol Hwan, Cho, Suk Young, Skene, Robert, Yamamoto, Syunsuke, Satou, Yousuke, Kuno, Masako, Miyazaki, Takahiro, Nakagawa, Hideyuki, Okabe, Atsutoshi, Marui, Shogo, Aso, Kazuyoshi, Yoshida, Masato
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cited_by cdi_FETCH-LOGICAL-c967-af22385b44768371ff93b5af081eea49b6f267588a3536da8df3e15574ca09de3
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container_end_page 749
container_issue 2
container_start_page 733
container_title Journal of medicinal chemistry
container_volume 59
creator Yogo, Takatoshi
Nagamiya, Hiroyuki
Seto, Masaki
Sasaki, Satoshi
Shih-Chung, Huang
Ohba, Yusuke
Tokunaga, Norihito
Lee, Gil Nam
Rhim, Chul Yun
Yoon, Cheol Hwan
Cho, Suk Young
Skene, Robert
Yamamoto, Syunsuke
Satou, Yousuke
Kuno, Masako
Miyazaki, Takahiro
Nakagawa, Hideyuki
Okabe, Atsutoshi
Marui, Shogo
Aso, Kazuyoshi
Yoshida, Masato
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doi_str_mv 10.1021/acs.jmedchem.5b01857
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title Structure-Based Design and Synthesis of 3-Amino-1,5-dihydro-4 H -pyrazolopyridin-4-one Derivatives as Tyrosine Kinase 2 Inhibitors
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