Electrogenerated base-promoted synthesis and antimicrobial activity of 2-imino-1,3-thiazolidin-4-one derivatives

Electrogenerated cyanomethylanions obtained by reduction of dry acetonitrile at a steel grid cathode were used to promote the addition of ethyl bromoacetate to thiourea derivatives. The reaction yields the corresponding 2-imino-1,3-thiazolidin-4-one. The reaction pathway was discussed based on the k...

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Published in:Journal of sulfur chemistry 2016-07, Vol.37 (4), p.391-400
Main Authors: Haouas, Beya, Saied, Taieb, Ayari, Hanen, Arfaoui, Youssef, Benkhoud, Mohamed Lamine, Boujlel, Khaled
Format: Article
Language:English
Subjects:
acetonitrile
antimicrobial activity
Antimicrobial agents
electrogenerated base
thiazolidinone
Thiourea
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description Electrogenerated cyanomethylanions obtained by reduction of dry acetonitrile at a steel grid cathode were used to promote the addition of ethyl bromoacetate to thiourea derivatives. The reaction yields the corresponding 2-imino-1,3-thiazolidin-4-one. The reaction pathway was discussed based on the kinetic and thermodynamic data obtained by computational methods. In addition, the biological activity of these new compounds was also investigated.
doi_str_mv 10.1080/17415993.2016.1155588
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subjects acetonitrile
antimicrobial activity
Antimicrobial agents
electrogenerated base
thiazolidinone
Thiourea
title Electrogenerated base-promoted synthesis and antimicrobial activity of 2-imino-1,3-thiazolidin-4-one derivatives
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