Chan-Lam-Evans Coupling of Cbz-Protected Histidines

Direct functionalization of protected histidines with arylboronic acids is described under Chan–Lam–Evans conditions to give the corresponding N(τ)‐arylhistidines in moderate to good yields (12 examples, up to 83 % yield) under mild conditions. Direct functionalization of protectedhistidines with ar...

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Bibliographic Details
Published in:European Journal of Organic Chemistry 2010-07, Vol.2010 (20), p.3811-3814
Main Authors: DalZotto, Christophe, Michaux, Julien, Martinand-Lurin, Elodie, Campagne, Jean-Marc
Format: Article
Language:English
Subjects:
Amino acids
Chemical Sciences
Chemistry
Copper
Cross-coupling
Exact sciences and technology
Heterocyclic compounds
Heterocyclic compounds with several n hetero atoms in the same ring, in separated rings or in fused rings
Organic chemistry
Peptides
Peptidomimetics
Preparations and properties
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Summary:Direct functionalization of protected histidines with arylboronic acids is described under Chan–Lam–Evans conditions to give the corresponding N(τ)‐arylhistidines in moderate to good yields (12 examples, up to 83 % yield) under mild conditions. Direct functionalization of protectedhistidines with arylboronic acids is described under Chan–Lam–Evans conditions to give the corresponding N(τ)‐arylhistidines in moderate to good yields (12 examples, up to 83 % yield) under mild conditions.
ISSN:1434-193X
1099-0690
DOI:10.1002/ejoc.201000591