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5-chloro-N-(4-methoxy-3-piperazin-1-yl-phenyl)-3-methyl-2-benzothiophenesulfonamide (SB-271046) : A potent, selective, and orally bioavailable 5-HT6 receptor antagonist

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Published in:	Journal of medicinal chemistry 1999-01, Vol.42 (2), p.202-205
Main Authors:	BROMIDGE, S. M, BROWN, A. M, MOSS, S. F, NEWMAN, H, RILEY, G, ROUTLEDGE, C, WYMAN, P, CLARKE, S. E, DODGSON, K, GAGER, T, GRASSAM, H. L, JEFFREY, P. M, JOINER, G. F, KING, F. D, MIDDLEMISS, D. N
Format:	Article
Language:	English
Subjects:	Biological and medical sciences Medical sciences Neuropharmacology Neurotransmitters. Neurotransmission. Receptors Pharmacology. Drug treatments Serotoninergic system
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container_title	Journal of medicinal chemistry
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creator	BROMIDGE, S. M BROWN, A. M MOSS, S. F NEWMAN, H RILEY, G ROUTLEDGE, C WYMAN, P CLARKE, S. E DODGSON, K GAGER, T GRASSAM, H. L JEFFREY, P. M JOINER, G. F KING, F. D MIDDLEMISS, D. N
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doi_str_mv	10.1021/jm980532e
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source	American Chemical Society:Jisc Collections:American Chemical Society Read & Publish Agreement 2022-2024 (Reading list)
subjects	Biological and medical sciences Medical sciences Neuropharmacology Neurotransmitters. Neurotransmission. Receptors Pharmacology. Drug treatments Serotoninergic system
title	5-chloro-N-(4-methoxy-3-piperazin-1-yl-phenyl)-3-methyl-2-benzothiophenesulfonamide (SB-271046) : A potent, selective, and orally bioavailable 5-HT6 receptor antagonist
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