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Pharmacokinetics and metabolism studies on 3-tert-butyl-7-(5-methylisoxazol-3-yl)-2-(1-methyl-1H-1,2,4-triazol-5-ylmethoxy) pyrazolo[1,5-d][1,2,4]triazine, a functionally selective GABAA α5 inverse agonist for cognitive dysfunction

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Published in:Bioorganic & medicinal chemistry letters 2006, Vol.16 (4), p.872-875
Main Authors: JONES, Philip, ATACK, John R, SZETO, Nicola, WAFFORD, Keith A, MACLEOD, Angus M, BRAUN, Matthew P, CATO, Brian P, CHAMBERS, Mark S, O'CONNOR, Desmond, COOK, Susan M, HOBBS, Sarah C, MAXEY, Robert, SZEKERES, Helen J
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container_issue 4
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container_title Bioorganic & medicinal chemistry letters
container_volume 16
creator JONES, Philip
ATACK, John R
SZETO, Nicola
WAFFORD, Keith A
MACLEOD, Angus M
BRAUN, Matthew P
CATO, Brian P
CHAMBERS, Mark S
O'CONNOR, Desmond
COOK, Susan M
HOBBS, Sarah C
MAXEY, Robert
SZEKERES, Helen J
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1464-3405
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source Elsevier
subjects Biological and medical sciences
Contrast media. Radiopharmaceuticals
Gabaergic and benzodiazepinic system
Medical sciences
Neuropharmacology
Neurotransmitters. Neurotransmission. Receptors
Pharmacology. Drug treatments
title Pharmacokinetics and metabolism studies on 3-tert-butyl-7-(5-methylisoxazol-3-yl)-2-(1-methyl-1H-1,2,4-triazol-5-ylmethoxy) pyrazolo[1,5-d][1,2,4]triazine, a functionally selective GABAA α5 inverse agonist for cognitive dysfunction
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