Cross-Coupling Reactions of Pyrimidin-2-yl Sulfonates with Phenols and Anilines： An Efficient Approach to C2-Functionalized Pyrimidines

Pyrimidin-2-yl sulfonates, as an efficient reaction partner, which can be easily prepared from cheap commercial materials, were coupled with phenols and anilines to give a wide array of C2-aryloxy- and arylaminopyrimidines in good to excellent yields under mild reaction conditions.

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Bibliographic Details
Published in:Chinese journal of chemistry 2013-12, Vol.31 (12), p.1495-1502
Main Authors: Quan, Zhengjun, Jing, Fuqiang, Zhang, Zhang, Da, Yuxia, Wang, Xicun
Format: Article
Language:English
Subjects:
C2-arylaminopyrimidines
C2-aryloxypyrimidines
cross-coupling
Phenols
pyrimindine-2-yl sulfonates
交叉偶联反应
化合物
反应条件
嘧啶
磺酰基
磺酸盐
苯胺类
苯酚
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Description
Summary:Pyrimidin-2-yl sulfonates, as an efficient reaction partner, which can be easily prepared from cheap commercial materials, were coupled with phenols and anilines to give a wide array of C2-aryloxy- and arylaminopyrimidines in good to excellent yields under mild reaction conditions.
ISSN:1001-604X
1614-7065
DOI:10.1002/cjoc.201300536