One-Pot Synthesis of N-Arylpyrazoles from Arylhalides

A simple one-pot method for the synthesis of diversely functionalized pyrazoles from aryl nucleophiles, di-tert-butylazodicarboxlate, and 1,3-dicarbonyl or equivalent compounds is presented.

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Bibliographic Details
Published in:Organic letters 2009-05, Vol.11 (10), p.2097-2100
Main Authors: Gerstenberger, Brian S, Rauckhorst, Mark R, Starr, Jeremy T
Format: Article
Language:English
Subjects:
Catalysis
Combinatorial Chemistry Techniques
Hydrocarbons, Halogenated - chemistry
Molecular Structure
Pyrazoles - chemical synthesis
Pyrazoles - chemistry
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Description
Summary:A simple one-pot method for the synthesis of diversely functionalized pyrazoles from aryl nucleophiles, di-tert-butylazodicarboxlate, and 1,3-dicarbonyl or equivalent compounds is presented.
ISSN:1523-7060
1523-7052
DOI:10.1021/ol900515a