A New Paclitaxel Photoaffinity Analog with a 3-(4-Benzoylphenyl)propanoyl Probe for Characterization of Drug-Binding Sites on Tubulin and P-Glycoprotein

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Published in:Journal of medicinal chemistry 1995-09, Vol.38 (20), p.3891-3894
Main Authors: Ojima, Iwao, Duclos, Olivier, Dorman, Gyorgy, Simonot, Bruno, Prestwich, Glenn D, Rao, Srinivasa, Lerro, Keith A, Horwitz, Susan B
Format: Article
Language:English
Subjects:
Affinity Labels - metabolism
Animals
Antineoplastic agents
Antineoplastic Agents - metabolism
ATP Binding Cassette Transporter, Subfamily B, Member 1 - metabolism
Binding Sites
Biological and medical sciences
General aspects
Medical sciences
Mice
Paclitaxel - analogs & derivatives
Paclitaxel - metabolism
Pharmacology. Drug treatments
Taxoids
Tubulin - metabolism
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cited_by cdi_FETCH-LOGICAL-a383t-407753aae6e8f91ebfb3917476d034b6f01428390db53d0b8698c0b1aec55a533
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container_end_page 3894
container_issue 20
container_start_page 3891
container_title Journal of medicinal chemistry
container_volume 38
creator Ojima, Iwao
Duclos, Olivier
Dorman, Gyorgy
Simonot, Bruno
Prestwich, Glenn D
Rao, Srinivasa
Lerro, Keith A
Horwitz, Susan B
description
doi_str_mv 10.1021/jm00020a001
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ispartof Journal of medicinal chemistry, 1995-09, Vol.38 (20), p.3891-3894
issn 0022-2623
1520-4804
language eng
recordid cdi_proquest_miscellaneous_77534855
source ACS CRKN Legacy Archives
subjects Affinity Labels - metabolism
Animals
Antineoplastic agents
Antineoplastic Agents - metabolism
ATP Binding Cassette Transporter, Subfamily B, Member 1 - metabolism
Binding Sites
Biological and medical sciences
General aspects
Medical sciences
Mice
Paclitaxel - analogs & derivatives
Paclitaxel - metabolism
Pharmacology. Drug treatments
Taxoids
Tubulin - metabolism
title A New Paclitaxel Photoaffinity Analog with a 3-(4-Benzoylphenyl)propanoyl Probe for Characterization of Drug-Binding Sites on Tubulin and P-Glycoprotein
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