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Efficient synthesis of new 3-heteroaryl-1-functionalized 1H-indazoles
The efficient synthesis of novel 3-heteroaryl N-1-functionalized indazoles, via palladium cross-coupling reactions of ethyl (3-iodo-1H-indazol-1-yl)acetate with 2- and 3-pyrrolylboronic acids, 2-, 4- and 5-thiazolylstannanes, and other heteroarylmetallated derivatives are reported.
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| Published in: | Tetrahedron 2011-01, Vol.67 (1), p.100-105 |
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| Main Authors: | , , , , |
| Format: | Article |
| Language: | English |
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| cited_by | cdi_FETCH-LOGICAL-c332t-d9e091cd4ef7cfdc2a0f9074cdd45ac4353edd759de4f2d0eeb71d811051bd9d3 |
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| cites | cdi_FETCH-LOGICAL-c332t-d9e091cd4ef7cfdc2a0f9074cdd45ac4353edd759de4f2d0eeb71d811051bd9d3 |
| container_end_page | 105 |
| container_issue | 1 |
| container_start_page | 100 |
| container_title | Tetrahedron |
| container_volume | 67 |
| creator | Fraile, Alberto Martín, M. Rosario García Ruano, José Luis Díaz, Juan Antonio Arranz, Esther |
| description | The efficient synthesis of novel 3-heteroaryl N-1-functionalized indazoles, via palladium cross-coupling reactions of ethyl (3-iodo-1H-indazol-1-yl)acetate with 2- and 3-pyrrolylboronic acids, 2-, 4- and 5-thiazolylstannanes, and other heteroarylmetallated derivatives are reported. |
| doi_str_mv | 10.1016/j.tet.2010.11.021 |
| format | article |
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| ispartof | Tetrahedron, 2011-01, Vol.67 (1), p.100-105 |
| issn | 0040-4020 1464-5416 |
| language | eng |
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| source | ScienceDirect Freedom Collection 2022-2024 |
| subjects | acetates azoles Chemical reactions Chemistry Derivatives Exact sciences and technology Heterocyclic compounds Heterocyclic compounds with n hetero atom and also o and/or s, se, te hetero atoms Heterocyclic compounds with only one n hetero atom and condensed derivatives Heterocyclic compounds with several n hetero atoms in the same ring, in separated rings or in fused rings Organic chemistry Palladium Preparations and properties synthesis Synthesis (chemistry) Tetrahedrons |
| title | Efficient synthesis of new 3-heteroaryl-1-functionalized 1H-indazoles |
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