Organocatalytic synthesis of benzazetidines by trapping hemiaminals with protecting groups

Benzazetidines are highly strained and inherently unstable heterocycles. There are only few methodologies for assem-bling these compounds. Here, a protocol is presented to trap an elusive cyclic, 4-membered hemiaminal structure. This method affords several benzazetidine in moderate to good yields (u...

Full description

Bibliographic Details

Main Authors:	Riccardo Salvio, Simone Placidi, Arianna Sinibaldi, Antonio Di Sabato, Dario C. Buscemi, Andrea Rossi, Achille Antenucci, Andrei Malkov, M. Bella
Format:	Default Article
Published:	2019
Subjects:	Organic chemistry not elsewhere classified Other chemical sciences not elsewhere classified Hemiaminals Benzazetidine Ring strain Strained heterocycles Chemical Sciences not elsewhere classified Organic Chemistry
Online Access:	https://hdl.handle.net/2134/37863
Tags:	Add Tag No Tags, Be the first to tag this record!